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FDA Established Pharmacologic Classes

Drug classes

307 FDA pharmacologic classes, each with its medicines, generics and pharmacy prices (FDA NDC Directory, October 8, 2026).

Every class

5-alpha reductase inhibitors
3 medicines; FDA: 5-alpha Reductase Inhibitor
ACE inhibitors
19 medicines; FDA: Angiotensin Converting Enzyme Inhibitor
Aldosterone antagonists
3 medicines; FDA: Aldosterone Antagonist
Alkaloid
2 medicines
Alkylating Drug
16 medicines
Alpha blockers
10 medicines; FDA: alpha-Adrenergic Blocker
Amino Acid
11 medicines
Aminoketone
3 medicines
Aminosalicylate
4 medicines
Androgens
3 medicines; FDA: Androgen
Anthelmintic
4 medicines
Anti-coagulant
25 medicines
Anti-seizure medicines
14 medicines; FDA: Anti-epileptic Agent
Antiarrhythmic
17 medicines
Anticholinergics
24 medicines; FDA: Anticholinergic
Antidiarrheal
3 medicines
Antidote
3 medicines
Antiemetic
2 medicines
Antihistamines
4 medicines; FDA: Antihistamine
Antihistamines (H1 blockers)
22 medicines; FDA: Histamine-1 Receptor Antagonist
Antimalarial
8 medicines
Antimetabolite
3 medicines
Antiprotozoal
7 medicines
Antithyroid medicines
2 medicines; FDA: Thyroid Hormone Synthesis Inhibitor
ARBs (angiotensin II receptor blockers)
22 medicines; FDA: Angiotensin 2 Receptor Blocker
Aromatase inhibitors
3 medicines; FDA: Aromatase Inhibitor
Atypical antipsychotics
17 medicines; FDA: Atypical Antipsychotic
Azole antifungals
20 medicines; FDA: Azole Antifungal
Barbiturates
6 medicines; FDA: Barbiturate
Benzodiazepines
16 medicines; FDA: Benzodiazepine
Beta blockers
21 medicines; FDA: beta-Adrenergic Blocker
Beta-2 agonists (bronchodilators)
18 medicines; FDA: beta2-Adrenergic Agonist
Biguanides (metformin)
13 medicines; FDA: Biguanide
Bile Acid
3 medicines
Bisphosphonates
6 medicines; FDA: Bisphosphonate
Calcium channel blockers
12 medicines; FDA: Calcium Channel Blocker
Calcium channel blockers (dihydropyridines)
16 medicines; FDA: Dihydropyridine Calcium Channel Blocker
Catecholamine
7 medicines
Cephalosporins
21 medicines; FDA: Cephalosporin Antibacterial
Cholinesterase inhibitors
8 medicines; FDA: Cholinesterase Inhibitor
Corticosteroids
55 medicines; FDA: Corticosteroid
Diagnostic Dye
5 medicines
Direct thrombin inhibitors
3 medicines; FDA: Direct Thrombin Inhibitor
DPP-4 inhibitors
12 medicines; FDA: Dipeptidyl Peptidase 4 Inhibitor
Endoglycosidase
11 medicines
Ergot Derivative
3 medicines
Estrogens
15 medicines; FDA: Estrogen
Expectorant
4 medicines
Factor Xa inhibitors
4 medicines; FDA: Factor Xa Inhibitor
Fluoroquinolones
6 medicines; FDA: Fluoroquinolone Antibacterial
Folate Analog
2 medicines
Glinide
2 medicines
GLP-1 receptor agonists
8 medicines; FDA: GLP-1 Receptor Agonist
Gonadotropin
2 medicines
H2 blockers
6 medicines; FDA: Histamine-2 Receptor Antagonist
Insulin Analog
9 medicines
Interferon beta
2 medicines
Iron Chelator
3 medicines
Kinase inhibitors
73 medicines; FDA: Kinase Inhibitor
Lead Chelator
3 medicines
Leukotriene receptor antagonists
2 medicines; FDA: Leukotriene Receptor Antagonist
Lipid Emulsion
4 medicines
Loop diuretics
4 medicines; FDA: Loop Diuretic
Macrolide
2 medicines
Macrolides
4 medicines; FDA: Macrolide Antimicrobial
MAO inhibitors
5 medicines; FDA: Monoamine Oxidase Inhibitor
Menin Inhibitor
2 medicines
Methylxanthine
11 medicines
Mood Stabilizer
5 medicines
Muscle relaxants
7 medicines; FDA: Muscle Relaxant
NSAIDs (nonsteroidal anti-inflammatory drugs)
44 medicines; FDA: Nonsteroidal Anti-inflammatory Drug
Opioid antagonists
11 medicines; FDA: Opioid Antagonist
Opioids (opioid agonists)
30 medicines; FDA: Opioid Agonist
Osmotic Diuretic
2 medicines
Osmotic Laxative
50 medicines
P2Y12 inhibitors (antiplatelets)
4 medicines; FDA: P2Y12 Platelet Inhibitor
Partial opioid agonists
2 medicines; FDA: Partial Opioid Agonist
PCSK9 inhibitors
2 medicines; FDA: PCSK9 Inhibitor
PDE5 inhibitors
5 medicines; FDA: Phosphodiesterase 5 Inhibitor
Pediculicide
2 medicines
Penicillins
13 medicines; FDA: Penicillin-class Antibacterial
Phenothiazine
12 medicines
Phosphate Binder
29 medicines
Potassium Binder
2 medicines
Potassium Salt
32 medicines
Progestins
16 medicines; FDA: Progestin
Proton pump inhibitors (PPIs)
9 medicines; FDA: Proton Pump Inhibitor
Retinoid
15 medicines
Sclerosing Agent
2 medicines
SGLT2 inhibitors
11 medicines; FDA: Sodium-Glucose Cotransporter 2 Inhibitor
Sigma-1 Agonist
7 medicines
SNRIs (serotonin and norepinephrine reuptake inhibitors)
5 medicines; FDA: Serotonin and Norepinephrine Reuptake Inhibitor
Statins
9 medicines; FDA: HMG-CoA Reductase Inhibitor
Stimulants
17 medicines; FDA: Central Nervous System Stimulant
Sulfonylureas
6 medicines; FDA: Sulfonylurea
Surfactant
3 medicines
Tetracyclines
3 medicines; FDA: Tetracycline-class Drug
Thiazide diuretics
21 medicines; FDA: Thiazide Diuretic
Thiazide-like diuretics
6 medicines; FDA: Thiazide-like Diuretic
Thiazolidinediones
4 medicines; FDA: Thiazolidinedione
TNF blockers
7 medicines; FDA: Tumor Necrosis Factor Blocker
Tricyclic antidepressants
11 medicines; FDA: Tricyclic Antidepressant
Triptans
9 medicines; FDA: Serotonin-1b and Serotonin-1d Receptor Agonist
Typical antipsychotics
4 medicines; FDA: Typical Antipsychotic
Vasoconstrictor
2 medicines
Vasodilator
2 medicines
Vinca Alkaloid
3 medicines
Vitamin B12
3 medicines
Vitamin C
4 medicines
Vitamin D
3 medicines
Vitamin D Analog
3 medicines
Vitamin K
3 medicines
Xanthine oxidase inhibitors
2 medicines; FDA: Xanthine Oxidase Inhibitor

Source: FDA NDC Directory (pharmacologic classes) via openFDA