Bempedoic Acid/Ezetimibe and Cyclosporine Interaction

Drug interaction information between Bempedoic Acid/Ezetimibe and Cyclosporine.

Bempedoic Acid/Ezetimibe and Cyclosporine have a documented minor interaction in FDA labeling.

FDA drug labeling documents a minor-severity interaction between Bempedoic Acid/Ezetimibe and Cyclosporine. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Bempedoic Acid/Ezetimibe

ACL Inhibitor / Cholesterol Absorption Inhibitor

Drug B

Cyclosporine

Calcineurin Inhibitor (Immunosuppressant)

How They Interact

These drugs interact in a way that increases the concentration of both medicines in your system.

FDA Label Information

Cyclosporine Clinical Impact: Concomitant use of NEXLIZET and cyclosporine increases ezetimibe and cyclosporine concentrations. Intervention: Monitor cyclosporine concentrations in patients receiving NEXLIZET and cyclosporine. In patients treated with cyclosporine, weigh the potential effects of the increased exposure to ezetimibe from concomitant use against the benefits of alterations in lipid levels provided by NEXLIZET.

Bempedoic Acid/Ezetimibe Also Interacts With

View all Bempedoic Acid/Ezetimibe interactions →

Frequently Asked Questions

What SPL severity band is on file for Bempedoic Acid/Ezetimibe + Cyclosporine?

Compiled FDA labeling labels this pair minor. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Cyclosporine has 89 labeled pairs on file vs Bempedoic Acid/Ezetimibe's 7. In the minor band specifically: Bempedoic Acid/Ezetimibe has 3 (also Ezetimibe, Cholestyramine); Cyclosporine has 60 (also Adalimumab, Amiodarone, Amlodipine, Anidulafungin).

What mechanism field is on file for Bempedoic Acid/Ezetimibe and Cyclosporine?

These drugs interact in a way that increases the concentration of both medicines in your system.

Cyclosporine carries more major-labeled pairs than Bempedoic Acid/Ezetimibe

SPL source-record counts only. This page's band is minor · classes on file: Bempedoic Acid/Ezetimibe (ACL Inhibitor / Cholesterol Absorption Inhibitor); Cyclosporine (Calcineurin Inhibitor (Immunosuppressant)).

Cyclosporine has 5 major-labeled pairs vs Bempedoic Acid/Ezetimibe's 0. This page itself is in the minor band, not the major band.

Bempedoic Acid/Ezetimibe

0 major · 4 moderate · 3 minor · 7 total

Cyclosporine

5 major · 24 moderate · 60 minor · 89 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.