Bempedoic Acid/Ezetimibe and Bempedoic Acid Interaction

Drug interaction information between Bempedoic Acid/Ezetimibe and Bempedoic Acid.

Bempedoic Acid/Ezetimibe and Bempedoic Acid have a documented moderate interaction in FDA labeling.

FDA drug labeling documents a moderate-severity interaction between Bempedoic Acid/Ezetimibe and Bempedoic Acid. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Bempedoic Acid/Ezetimibe

ACL Inhibitor / Cholesterol Absorption Inhibitor

Drug B

Bempedoic Acid

ACL Inhibitor

How They Interact

This combination can cause simvastatin levels to build up in your body, which increases the risk of muscle damage.

FDA Label Information

7 DRUG INTERACTIONS No specific pharmacokinetic drug interaction studies with NEXLIZET have been conducted. Table 4 lists drug interactions with NEXLIZET that have been identified in studies with bempedoic acid or ezetimibe. Clinically Important Drug Interactions with NEXLIZET Simvastatin Clinical Impact: Concomitant use of NEXLIZET with simvastatin causes an increase in simvastatin concentration and may increase the risk of simvastatin-related myopathy [see Clinical Pharmacology (12.3) ] .

Bempedoic Acid/Ezetimibe Also Interacts With

View all Bempedoic Acid/Ezetimibe interactions →

Frequently Asked Questions

What SPL severity band is on file for Bempedoic Acid/Ezetimibe + Bempedoic Acid?

Compiled FDA labeling labels this pair moderate. That is a source-record field, not an individual medication-combination decision.

How many labeled pairs sit in each drug's moderate band?

Bempedoic Acid/Ezetimibe and Bempedoic Acid tie at 7 labeled pairs each. moderate-band counts: Bempedoic Acid/Ezetimibe 4 alongside Simvastatin, Pravastatin, Fenofibrate; Bempedoic Acid 4 alongside Simvastatin, Pravastatin, Fenofibrate.

What mechanism field is on file for Bempedoic Acid/Ezetimibe and Bempedoic Acid?

This combination can cause simvastatin levels to build up in your body, which increases the risk of muscle damage.

Bempedoic Acid/Ezetimibe and Bempedoic Acid · moderate-band peers

SPL source-record counts only. This page's band is moderate · classes on file: Bempedoic Acid/Ezetimibe (ACL Inhibitor / Cholesterol Absorption Inhibitor); Bempedoic Acid (ACL Inhibitor).

Bempedoic Acid/Ezetimibe

0 major · 4 moderate · 3 minor · 7 total

Bempedoic Acid

0 major · 4 moderate · 3 minor · 7 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.