Phenelzine and Sertraline Interaction

Drug interaction information between Phenelzine and Sertraline.

Phenelzine and Sertraline have a documented moderate interaction in FDA labeling.

FDA drug labeling documents a moderate-severity interaction between Phenelzine and Sertraline. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Phenelzine

Monoamine Oxidase Inhibitor (MAOI)

Drug B

Sertraline

Selective Serotonin Reuptake Inhibitor (SSRI)

How They Interact

Both of these drugs increase a chemical in your brain called serotonin. Taking them together can cause dangerously high levels of serotonin, which can be life-threatening.

FDA Label Information

Drug Interactions In patients receiving nonselective monoamine oxidase (MAO) inhibitors in combination with serotoninergic agents (e.g., dexfenfluramine, fluoxetine, fluvoxamine, paroxetine, sertraline, citalopram, venlafaxine) there have been reports of serious, sometimes fatal, reactions.

Phenelzine Also Interacts With

View all Phenelzine interactions →

Frequently Asked Questions

What SPL severity band is on file for Phenelzine + Sertraline?

Compiled FDA labeling labels this pair moderate. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Sertraline has 34 labeled pairs on file vs Phenelzine's 27. In the moderate band specifically: Phenelzine has 11 (also Fluoxetine, Citalopram, Venlafaxine, Fluvoxamine); Sertraline has 2 (also Aspirin).

What mechanism field is on file for Phenelzine and Sertraline?

Both of these drugs increase a chemical in your brain called serotonin. Taking them together can cause dangerously high levels of serotonin, which can be life-threatening.

Sertraline carries more major-labeled pairs than Phenelzine

SPL source-record counts only. This page's band is moderate · classes on file: Phenelzine (Monoamine Oxidase Inhibitor (MAOI)); Sertraline (Selective Serotonin Reuptake Inhibitor (SSRI)).

Sertraline has 1 major-labeled pair vs Phenelzine's 0. This page itself is in the moderate band, not the major band.

Phenelzine

0 major · 11 moderate · 16 minor · 27 total

Sertraline

1 major · 2 moderate · 31 minor · 34 total

  • Other moderate peers for Sertraline
  • Aspirin

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.