Trazodone and Linezolid Interaction

Drug interaction information between Trazodone and Linezolid.

Trazodone and Linezolid have a documented major interaction in FDA labeling.

FDA drug labeling documents a major-severity interaction between Trazodone and Linezolid. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Trazodone

Serotonin Antagonist and Reuptake Inhibitor (SARI)

Drug B

Linezolid

Oxazolidinone Antibiotic

How They Interact

Linezolid acts like a special type of medicine that can cause a dangerous buildup of a brain chemical called serotonin when mixed with trazodone. This can lead to a serious condition called serotonin syndrome.

FDA Label Information

Intervention: Trazodone is contraindicated in patients taking MAOIs, including MAOIs such as linezolid or intravenous methylene blue [see Contraindications (4), Dosage and Administration (2.3, 2.4), and Warnings and Precautions (5.2)].

Trazodone Also Interacts With

View all Trazodone interactions →

Frequently Asked Questions

What SPL severity band is on file for Trazodone + Linezolid?

Compiled FDA labeling labels this pair major. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Trazodone has 40 labeled pairs on file vs Linezolid's 29. In the major band specifically: Trazodone has 1; Linezolid has 8 (also Citalopram, Escitalopram, Mirtazapine, Paroxetine).

What mechanism field is on file for Trazodone and Linezolid?

Linezolid acts like a special type of medicine that can cause a dangerous buildup of a brain chemical called serotonin when mixed with trazodone. This can lead to a serious condition called serotonin syndrome.

Linezolid carries more major-labeled pairs than Trazodone

SPL source-record counts only. This page's band is major · classes on file: Trazodone (Serotonin Antagonist and Reuptake Inhibitor (SARI)); Linezolid (Oxazolidinone Antibiotic).

Linezolid has 8 major-labeled pairs vs Trazodone's 1.

Trazodone

1 major · 4 moderate · 35 minor · 40 total

Trazodone has no other major-band peer in this dataset besides Linezolid.

Linezolid

8 major · 3 moderate · 18 minor · 29 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.