Spironolactone and Cholestyramine Interaction

Drug interaction information between Spironolactone and Cholestyramine.

Spironolactone and Cholestyramine have a documented minor interaction in FDA labeling.

FDA drug labeling documents a minor-severity interaction between Spironolactone and Cholestyramine. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Spironolactone

Anti-Androgen

Drug B

Cholestyramine

Bile Acid Sequestrant

How They Interact

Using these medicines at the same time can cause your blood to become too acidic and hold onto too much potassium.

FDA Label Information

• Cholestyramine: Hyperkalemic metabolic acidosis has been reported with concomitant use ( 7.5 ). 7.5 Cholestyramine Hyperkalemic metabolic acidosis has been reported in patients given ALDACTONE concurrently with cholestyramine.

Spironolactone Also Interacts With

View all Spironolactone interactions →

Cholestyramine Also Interacts With

View all Cholestyramine interactions →

Frequently Asked Questions

What SPL severity band is on file for Spironolactone (Acne) + Cholestyramine?

Compiled FDA labeling labels this pair minor. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Cholestyramine has 34 labeled pairs on file vs Spironolactone's 7. In the minor band specifically: Spironolactone has 3 (also Spironolactone, Digoxin); Cholestyramine has 31 (also Propranolol, Warfarin, Tetracycline, Phenobarbital).

What mechanism field is on file for Spironolactone (Acne) and Cholestyramine?

Using these medicines at the same time can cause your blood to become too acidic and hold onto too much potassium.

Cholestyramine's labeled portfolio outnumbers Spironolactone

SPL source-record counts only. This page's band is minor · classes on file: Spironolactone (Anti-Androgen); Cholestyramine (Bile Acid Sequestrant).

Spironolactone

0 major · 4 moderate · 3 minor · 7 total

Cholestyramine

0 major · 3 moderate · 31 minor · 34 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.