Quetiapine and Itraconazole Interaction

Drug interaction information between Quetiapine and Itraconazole.

Quetiapine and Itraconazole have a documented minor interaction in FDA labeling.

FDA drug labeling documents a minor-severity interaction between Quetiapine and Itraconazole. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Quetiapine

Atypical Antipsychotic

Drug B

Itraconazole

Azole Antifungal

How They Interact

Itraconazole slows down how fast your body gets rid of quetiapine, which can cause the medicine to build up to high levels.

FDA Label Information

Quetiapine exposure is increased by the prototype CYP3A4 inhibitors (e.g., ketoconazole, itraconazole, indinavir, ritonavir, nefazodone, etc.) and decreased by the prototype CYP3A4 inducers (e.g., phenytoin, carbamazepine, rifampin, avasimibe, St.

Frequently Asked Questions

What SPL severity band is on file for Quetiapine + Itraconazole?

Compiled FDA labeling labels this pair minor. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Itraconazole has 116 labeled pairs on file vs Quetiapine's 9. In the minor band specifically: Quetiapine has 7 (also Ketoconazole, Carbamazepine, Rifampin, Dopamine); Itraconazole has 77 (also Fluticasone, Meloxicam, Buspirone, Oxycodone).

What mechanism field is on file for Quetiapine and Itraconazole?

Itraconazole slows down how fast your body gets rid of quetiapine, which can cause the medicine to build up to high levels.

Itraconazole carries more major-labeled pairs than Quetiapine

SPL source-record counts only. This page's band is minor · classes on file: Quetiapine (Atypical Antipsychotic); Itraconazole (Azole Antifungal).

Itraconazole has 19 major-labeled pairs vs Quetiapine's 1. This page itself is in the minor band, not the major band.

Quetiapine

1 major · 1 moderate · 7 minor · 9 total

Itraconazole

19 major · 20 moderate · 77 minor · 116 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.