Rifampin · more major-labeled pairs than Abiraterone

SPL labels Abiraterone + Rifampin as minor; Abiraterone 5 / Rifampin 103 in that band.

Mechanism on file: Rifampin makes your liver work faster to get rid of abiraterone. This lowers the amount of abiraterone in your blood, which could make it less effective.

FDA SPL severity: Minor

Abiraterone

Full Abiraterone label record

CYP17 Inhibitor

Rifampin

Full Rifampin label record

Rifamycin Antibiotic

Abiraterone + Rifampin · SPL mechanism field

Rifampin makes your liver work faster to get rid of abiraterone. This lowers the amount of abiraterone in your blood, which could make it less effective.

Minor band excerpt · Abiraterone with Rifampin

In a dedicated drug interaction trial, co-administration of rifampin, a strong CYP3A4 inducer, decreased exposure of abiraterone by 55%.

Rifampin · 8 major-labeled pairs (vs Abiraterone's 0)

View all Rifampin interactions →

FDA Drug Labels (SPL) via openFDA. Registry display only. Not medical advice.