Pioglitazone · more major-labeled pairs than Metformin/Pioglitazone

SPL labels Pioglitazone + Metformin/Pioglitazone as minor; Pioglitazone 9 / Metformin/Pioglitazone 7 in that band.

Mechanism on file: Other medications can change how your body processes pioglitazone, leading to levels that are either too high or too low.

FDA SPL severity: Minor

Pioglitazone

Full Pioglitazone label record

Thiazolidinedione

Metformin/Pioglitazone

Full Metformin/Pioglitazone label record

Biguanide / TZD Combination

Pioglitazone + Metformin/Pioglitazone · SPL mechanism field

Other medications can change how your body processes pioglitazone, leading to levels that are either too high or too low.

Minor band excerpt · Pioglitazone with Metformin/Pioglitazone

( 7.1 ) CYP2C8 inducers (e.g., rifampin) may decrease pioglitazone concentrations. ( 7.6 ) Topiramate may decrease pioglitazone concentrations. ( 7.8 ) 7.1 Strong CYP2C8 Inhibitors An inhibitor of CYP2C8 (e.g., gemfibrozil) significantly increases the exposure (area under the serum concentration-time curve or AUC) and half-life (t ½ ) of pioglitazone.

Pioglitazone · 1 major-labeled pairs (vs Metformin/Pioglitazone's 0)

View all Pioglitazone interactions →

Metformin/Pioglitazone · 7 minor + 10 total pairs

View all Metformin/Pioglitazone interactions →

FDA Drug Labels (SPL) via openFDA. Registry display only. Not medical advice.