Prescription medication · Anticonvulsant (GABA Reuptake Inhibitor)

tiagabine

Also sold as Gabitril. Tiagabine is used to treat partial seizures in adults and children 12 years and older.

Data updated 2026-05-15

81
FDA reportsRarely reported
11
InteractionsSeveral interactions
$5.41
Generic price (NADAC)

What the data shows

tiagabine (Gabitril) is a prescription Anticonvulsant (GABA Reuptake Inhibitor), among the least-reported drugs the FDA tracks (81 FDA reports), with 11 documented drug interactions.

Reporting volume reflects how widely a drug is used and studied, not how dangerous it is, a FAERS report documents a temporal association, never proof of cause.

tiagabine (Gabitril) is a prescription Anticonvulsant (GABA Reuptake Inhibitor). Tiagabine is used to treat partial seizures in adults and children 12 years and older.

Tiagabine is a medicine used with other medicines to treat partial seizures. It helps to control seizures by affecting certain chemicals in the brain.

Drug Pricing (NADAC)

Generic Price

$5.41/unit

Generic Available

Yes (2 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

Compare with Another Drug → Full Side Effects Report →

What it does

Tiagabine is used to treat partial seizures in adults and children 12 years and older.

Common side effects

Dizziness, Lack of energy, Sleepiness

Key warnings

This medicine may cause serious side effects.

The sections below are summarized in plain English from tiagabine's FDA-approved prescribing information. They describe what the official label says, and are not personal medical advice.

How It Works

Tiagabine works by increasing the amount of a chemical called GABA in the brain. GABA helps to calm the brain and reduce seizures. Tiagabine blocks the reuptake of GABA, which means more GABA is available in the brain.

Side Effects (from patient reports)

Based on 81 FDA adverse event reports.

Most-reported reactions

Adverse reactions in FAERS for tiagabine, by number of reports

reports

What this shows Bars show how often each reaction was reported, not how likely it is to happen, a report records a temporal association, never proof that the drug caused it.

Source FDA Adverse Event Reporting System (FAERS) As of 2025

Reports over time

Adverse-event reports filed for tiagabine each year to the FDA Adverse Event Reporting System (FAERS).

05101520 2004200720112014201920222025 6

Year-to-year volume tracks usage, prescribing, and scrutiny, not a change in per-patient risk. Source: FDA FAERS.

Where tiagabine sits

tiagabine has more FDA adverse-event reports than 1% of the drugs FAERS tracks. A high position reflects how widely a drug is used and watched, not how dangerous it is.

fewest reports most reports

Percentile across all drugs PlainMeds tracks by FAERS report volume. The dot is tiagabine; the line is the median (50th percentile).

FDA Adverse Event Report Analysis

Detailed analysis of 81 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2004–2025.

Total Reports

81

Reports Mentioning Death

7

8.6% of reports — not proof of cause

Hospitalization Reports

32

Top Indication

Multiple Sclerosis

Gender Distribution

Female 55 (76%)
Male 17 (24%)

Age Distribution

0–17 1
18–44 17
45–64 26
65–74 8
75+ 1

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 ENCEPHALOPATHY 16
2 MYOCLONUS 14
5 DIZZINESS 6
6 FEELING ABNORMAL 5
7 SEIZURE 5
9 SEROTONIN SYNDROME 4
10 TOXICITY TO VARIOUS AGENTS 4
11 TREMOR 4
12 ABNORMAL BEHAVIOUR 3
13 COMPLETED SUICIDE 3
14 DRUG INTERACTION 3
15 DYSKINESIA 3
16 FATIGUE 3
17 HEADACHE 3
18 INSOMNIA 3

Reactions in Death Reports

COMPLETED SUICIDE 3
DEATH 2
CARDIAC ARREST 1
CONVULSION 1
OVERDOSE 1
RESPIRATORY ARREST 1
UNEVALUABLE EVENT 1
WEIGHT INCREASED 1

Reactions in Hospitalization Reports

ENCEPHALOPATHY 14
MYOCLONUS 14
FATIGUE 3
INSOMNIA 3
TOXICITY TO VARIOUS AGENTS 3
ANXIETY 2
DRUG INTERACTION 2
DYSARTHRIA 2
DYSKINESIA 2
HAEMOGLOBIN DECREASED 2

Source: FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

This medicine may cause serious side effects. Tell your doctor right away if you have any changes in mood or behavior, or any suicidal thoughts.

Known Drug Interactions

Carbamazepine, phenytoin, primidone, and phenobarbital are generally classified as enzyme inducers; valproate and gabapentin are not.

Mechanism: Gabapentin does not speed up or slow down the liver enzymes that process tiagabine. This means it is unlikely to change how much tiagabine stays in your body.

Warfarin: No significant differences were observed in the steady-state pharmacokinetics of R-warfarin or S-warfarin with the addition of tiagabine given as a single dose.

Mechanism: Studies show that tiagabine does not change the levels of warfarin in the blood. The two drugs do not seem to have a meaningful interaction.

Carbamazepine, phenytoin, primidone, and phenobarbital are generally classified as enzyme inducers; valproate and gabapentin are not. Valproate: Tiagabine causes a slight decrease (about 10%) in steady-state valproate concentrations. Valproate: The addition of tiagabine to patients taking valproate chronically had no effect on tiagabine pharmacokinetics, but valproate significantly decreased tiagabine binding in vitro from 96.3 to 94.8%, which resulted in an increase of approximately 40% in the free tiagabine concentration.

Mechanism: Valproate pushes tiagabine off blood proteins, which increases the amount of active tiagabine in the body. Tiagabine also slightly lowers the levels of valproate.

minor digoxin

Digoxin: Concomitant administration of tiagabine did not affect the steady-state pharmacokinetics of digoxin or the mean daily trough serum level of digoxin.

Mechanism: These two drugs do not interfere with each other's levels or how the body uses them.

Theophylline: A single 10 mg dose of tiagabine did not affect the pharmacokinetics of theophylline at steady state.

Mechanism: Tiagabine does not change how the body breaks down or handles theophylline.

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This is a plain-language summary of FDA-label interaction records and does not provide individual medication-combination directions.

Common Questions

Can I stop taking tiagabine suddenly?
Do not stop taking tiagabine suddenly without talking to your doctor. Stopping suddenly can cause seizures.
Will tiagabine interact with my other medications?
Tiagabine can interact with other medications, especially other seizure medicines. Tell your doctor about all the medicines you take.
Can I drink alcohol while taking tiagabine?
Talk to your doctor about drinking alcohol while taking tiagabine. Alcohol can increase the risk of side effects.
How often will my dose be adjusted?
Your doctor may adjust your dose of tiagabine every week, depending on how well it is working and how you are tolerating it.
What should I do if I experience side effects?
Tell your doctor if you experience any side effects while taking tiagabine.
Is it safe to drive while taking tiagabine?
Tiagabine may cause drowsiness or dizziness. Do not drive or operate machinery until you know how tiagabine affects you.
Can children take tiagabine?
Tiagabine is approved for use in children 12 years and older.
What do I do if I accidentally take too much tiagabine?
Seek medical attention immediately.
Does food affect how tiagabine works?
Yes, you should take tiagabine with food.
How will I know if the medicine is working?
You should have fewer seizures.
What are the common side effects of tiagabine?
The registry lists Dizziness, Lack of energy, Sleepiness, Nausea, Nervousness or irritability among the most-reported FAERS reaction terms for tiagabine. The compiled record contains 81 FDA adverse-event reports. These counts are not an individual symptom assessment.
Does tiagabine interact with other medications?
The registry has 11 documented interaction rows for tiagabine. Notable source-record pairings include gabapentin, warfarin, valproate. These rows are not a complete medication review.
What drug class is tiagabine?
tiagabine belongs to the Anticonvulsant (GABA Reuptake Inhibitor) drug class. It requires a prescription (Rx). Tiagabine is used to treat partial seizures in adults and children 12 years and older.
What pregnancy or breastfeeding source fields are listed for tiagabine?
The FDA label for tiagabine contains product-specific pregnancy or breastfeeding language. PlainMeds does not apply that source text to an individual.

Other drugs grouped near tiagabine - same-class peers and common alternatives.

Compare tiagabine vs brivaracetam side-by-side →

Compare beyond drug class

Nationwide peers by FAERS volume & death-report share

Two PlainMeds-derived comparison paths for tiagabine: nearest FDA FAERS report volume and nearest death-report share among drugs with at least 1,000 logged reports, excluding same-class neighbors listed above. Counts reflect reporting volume, not proven individual harm.

Medication Guides

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What the FDA Data Shows for tiagabine

The FDA label for tiagabine (sold under brand names such as Gabitril) classifies it as a prescription-only medication in the Anticonvulsant (GABA Reuptake Inhibitor) class. Tiagabine is used to treat partial seizures in adults and children 12 years and older. Official labeling lists 8 commonly reported side effects, including Dizziness, Lack of energy, Sleepiness.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 81 voluntary reports. The database also lists 11 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated minor severity. NADAC pricing from CMS shows a generic unit cost of $5.41.

Report counts do not establish causation, a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information are separate source-record fields. This page is a public FDA/CMS registry and does not provide medical, treatment, substitution, or medication-change directions.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. This registry does not provide medication decisions.

Last updated: March 1, 2021

PlainMeds is rendered directly from FDA openFDA/FAERS extracts, DailyMed labels, and CMS drug-pricing files, no number is typed in by an editor. FAERS counts, recalls, shortages, and price figures on this page are queried live from those federal extracts. See our editorial standards & corrections policy, the methodology behind these numbers, or report a data error. Data current as of 2026-05-15. Primary sources: openFDA / FAERS, DailyMed and CMS Part B ASP.

Data currency: FDA FAERS adverse-event reports through 2025, CMS NADAC acquisition-cost pricing effective December 2024, compiled from the source snapshot dated . See our methodology for per-source dates and refresh cadence. Spot a figure that looks wrong? Report a data issue.

All federal data sources used on this page