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sulfasalazine

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Brand names: Azulfidine

Disease-Modifying Antirheumatic Drug (DMARD) Rx

Sulfasalazine is a drug that reduces inflammation in the body. It is used to treat ulcerative colitis.

Drug Pricing (NADAC)

Generic Price

$0.18/unit

Generic Available

Yes (5 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

Sulfasalazine treats ulcerative colitis, a condition that causes inflammation and sores in the lining of the large intestine.

Common side effects

Loss of appetite, Headache, Nausea

Key warnings

You should not take this medicine if you have a blockage in your intestines or urinary tract.

How It Works

Sulfasalazine is an anti-inflammatory drug. It works by reducing inflammation in the colon. The exact way it does this is not fully known.

How to Take It

Take Sulfasalazine as your doctor tells you. The usual starting dose for adults is 3 to 4 grams per day, divided into equal doses taken every 8 hours. Some people start with a lower dose, like 1 to 2 grams per day, to avoid stomach problems. Your doctor may adjust your dose based on how well the medicine works for you.

Pregnancy & Breastfeeding

Tell your doctor if you are pregnant or plan to become pregnant. It is not known if Sulfasalazine will harm your unborn baby. Talk to your doctor about the risks and benefits of taking this medicine while breastfeeding.

Missed Dose

If you miss a dose, take it as soon as you remember. If it is close to your next dose, skip the missed dose and continue with your regular schedule.

Storage

Store at room temperature between 59°F and 86°F.

Side Effects (from patient reports)

Based on 147,268 FDA adverse event reports.

The medicine is not working
29,013
Rheumatoid arthritis
19,190
Pain
15,658
Cannot tolerate the medicine
13,521
Joint pain
13,161
Tiredness
13,017
Swollen joint
12,481
Using the medicine for a different purpose
10,749
Skin rash
10,677
Stomach discomfort
9,801

FDA Adverse Event Report Analysis

Detailed analysis of 76,270 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2003–2025.

Total Reports

76,270

Death-Related Reports

6,629

Hospitalization Reports

20,613

Top Indication

Rheumatoid Arthritis

Gender Distribution

Female 52,098 (77%)
Male 15,843 (23%)

Age Distribution

0–17 1,085
18–44 12,906
45–64 20,646
65–74 8,320
75+ 4,155

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 DRUG INEFFECTIVE 29,013
2 RHEUMATOID ARTHRITIS 19,190
3 PAIN 15,658
4 DRUG INTOLERANCE 13,521
5 ARTHRALGIA 13,161
6 FATIGUE 13,017
7 JOINT SWELLING 12,481
8 OFF LABEL USE 10,749
9 RASH 10,678
10 ABDOMINAL DISCOMFORT 9,801
11 CONTRAINDICATED PRODUCT ADMINISTERED 9,454
12 CONDITION AGGRAVATED 9,374
13 ALOPECIA 9,277
14 ARTHROPATHY 9,001
15 SYNOVITIS 8,965

Reactions in Death Reports

RHEUMATOID ARTHRITIS 2,082
SYSTEMIC LUPUS ERYTHEMATOSUS 2,074
OFF LABEL USE 2,037
TYPE 2 DIABETES MELLITUS 2,028
JOINT SWELLING 1,999
SYNOVITIS 1,970
RASH 1,961
GLOSSODYNIA 1,958
WOUND 1,945
PSORIATIC ARTHROPATHY 1,939

Reactions in Hospitalization Reports

DRUG INEFFECTIVE 5,832
RHEUMATOID ARTHRITIS 5,015
PAIN 4,516
ARTHRALGIA 4,487
OFF LABEL USE 4,272
JOINT SWELLING 4,240
FATIGUE 4,179
RASH 3,909
DRUG INTOLERANCE 3,726
CONDITION AGGRAVATED 3,681

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

You should not take this medicine if you have a blockage in your intestines or urinary tract. You should not take this medicine if you have porphyria, as it could cause an attack. You should not take this medicine if you are allergic to sulfasalazine, its ingredients, sulfonamides, or salicylates.

Known Drug Interactions

Drugs That May Cause Methemoglobinemia When Used with LIDODERM Patients who are administered local anesthetics are at increased risk of developing methemoglobinemia when concurrently exposed to the following drugs, which could include other local anesthetics: Examples of Drugs Associated with Methemoglobinemia : Class Examples Nitrates/Nitrites nitric oxide, nitroglycerin, nitroprusside, nitrous oxide Local anesthetics articaine, benzocaine, bupivacaine, lidocaine, mepivacaine, prilocaine, procaine, ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, ifos...

Mechanism: Both drugs can cause a rare blood problem that prevents oxygen from reaching your body's tissues. Using them together makes this dangerous side effect more likely to happen.

What to do: Your doctor should monitor you closely for signs like blue skin or shortness of breath. Seek medical help immediately if you feel unusually tired or dizzy.

Coadministration of VOSEVI with BCRP substrates (e.g., methotrexate, mitoxantrone, imatinib, irinotecan, lapatinib, rosuvastatin, sulfasalazine, topotecan) is not recommended [see Clinical Pharmacology (12.3) ].

Mechanism: This medicine interferes with a protein that transports sulfasalazine, which could cause the levels of sulfasalazine in your body to rise.

What to do: The manufacturer does not recommend taking these two medications at the same time.

minor digoxin

John's Wort, sucralfate, sulfasalazine Measure serum digoxin concentrations before initiating concomitant drugs.

Mechanism: Sulfasalazine can decrease the amount of digoxin in your blood, making the heart medicine less effective.

What to do: Your doctor should check your digoxin levels before you begin taking this combination.

7.5 Effects of Other Drugs on Folates Several drugs have been reported to reduce folate concentrations by inhibition of the dihydrofolate reductase enzyme (e.g., methotrexate and sulfasalazine) or by reducing folate absorption (e.g., cholestyramine), or via unknown mechanisms (e.g., antiepileptics such as carbamazepine, phenytoin, phenobarbital, primidone and valproic acid).

Mechanism: Sulfasalazine can lower the levels of folate in your body by blocking a specific enzyme that helps process it.

What to do: Your doctor may need to monitor your folate levels or adjust your supplements while taking these medications together.

7.4 Sulfasalazine Patients in a clinical study who were on established therapy with sulfasalazine, to which Enbrel was added, were noted to develop a mild decrease in mean neutrophil counts in comparison to groups treated with either Enbrel or sulfasalazine alone.

Mechanism: Taking these two medicines together can lower the number of white blood cells that help your body fight infections.

What to do: Your doctor should monitor your blood cell counts regularly while you are using both medications.

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Common Questions

Can I take this with food?
The drug label does not specify whether to take it with food. Follow your doctor's instructions.
What if I have stomach upset?
If you have stomach upset, talk to your doctor. They may lower your dose or have you stop the medicine for a short time.
How long will I need to take this medicine?
You may need to continue taking this medicine even when your symptoms are under control. Talk to your doctor about how long you should take it.
Can this medicine affect my ability to have children?
Sulfasalazine can cause a reduced sperm count in men, which may be reversible when the drug is stopped.
What should I do if I think I'm having an allergic reaction?
Stop taking the medicine and seek immediate medical attention if you think you are having an allergic reaction.
Can I take other medicines with Sulfasalazine?
Tell your doctor about all the medicines you take, including prescription and over-the-counter drugs, vitamins, and herbal supplements.
Will this medicine cure my ulcerative colitis?
Sulfasalazine helps manage ulcerative colitis by reducing inflammation. It may not cure the condition, but it can help control symptoms and prevent flare-ups.
How long does it take for this medicine to work?
It may take several weeks or months to see the full effects of this medicine. Talk to your doctor if you don't notice any improvement in your symptoms.
Can this medicine cause my urine to change color?
Yes, Sulfasalazine can cause your urine to become discolored.
Is it safe to get vaccines while taking Sulfasalazine?
Talk to your doctor before getting any vaccines while taking Sulfasalazine.
What are the common side effects of sulfasalazine?
The most commonly reported side effects of sulfasalazine include Loss of appetite, Headache, Nausea, Vomiting, Stomach upset. Based on 147,268 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
Does sulfasalazine interact with other medications?
Yes, sulfasalazine has 7 known drug interactions. Notable interactions include lidocaine topical, sofosbuvir/velpatasvir, digoxin. Always inform your doctor about all medications you are taking.
What drug class is sulfasalazine?
sulfasalazine belongs to the Disease-Modifying Antirheumatic Drug (DMARD) drug class. It requires a prescription (Rx). Sulfasalazine treats ulcerative colitis, a condition that causes inflammation and sores in the lining of the large intestine.
Is sulfasalazine safe during pregnancy?
Tell your doctor if you are pregnant or plan to become pregnant. It is not known if Sulfasalazine will harm your unborn baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

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Related Health & Safety Data

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What the FDA Data Shows for sulfasalazine

The FDA label for sulfasalazine (sold under brand names such as Azulfidine) classifies it as a prescription-only medication in the Disease-Modifying Antirheumatic Drug (DMARD) class. Sulfasalazine treats ulcerative colitis, a condition that causes inflammation and sores in the lining of the large intestine. Official labeling lists 6 commonly reported side effects, including Loss of appetite, Headache, Nausea.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 147,268 voluntary reports. The database also lists 7 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated moderate severity. NADAC pricing from CMS shows a generic unit cost of $0.18.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: December 12, 2022

All federal data sources used on this page