Carbidopa/Levodopa · larger labeled portfolio than Entacapone

SPL labels Carbidopa/Levodopa + Entacapone as moderate; Carbidopa/Levodopa 8 / Entacapone 2 in that band.

Mechanism on file: Entacapone is designed to block the enzyme that breaks down levodopa, which helps the medicine stay in your system longer. This can increase the effects of the levodopa on your brain and body.

FDA SPL severity: Moderate

Carbidopa/Levodopa

Full Carbidopa/Levodopa label record

Dopamine Precursor Combination

Entacapone

Full Entacapone label record

COMT Inhibitor

Carbidopa/Levodopa + Entacapone · SPL mechanism field

Entacapone is designed to block the enzyme that breaks down levodopa, which helps the medicine stay in your system longer. This can increase the effects of the levodopa on your brain and body.

Moderate band excerpt · Carbidopa/Levodopa with Entacapone

7 DRUG INTERACTIONS Drugs metabolized by COMT: use with caution ( 5.10 , 7.2 ) Anti-hypertensive agents: dose adjustment may be required ( 7.3 ) Tricyclic antidepressants: risk of hypertension and dyskinesia reported during concomitant use with carbidopa/levodopa ( 7.4 ) Dopamine D2 receptor antagonists, isoniazid, phenytoin, papaverine and iron salts: may reduce efficacy of carbidopa, levodopa and entacapone tablets ( 7.5 , 7.6 , 7.7 , 7.8 , 7.9 ) Drugs that interfere with biliary excretion, glucuronidation and intestinal beta-glucuronidase: dose adjustment of carbidopa, levodopa and...

Carbidopa/Levodopa · 13 SPL pairs (broader portfolio than Entacapone)

View all Carbidopa/Levodopa interactions →

Entacapone · 2 moderate + 3 total pairs

View all Entacapone interactions →

FDA Drug Labels (SPL) via openFDA. Registry display only. Not medical advice.