Repaglinide · more major-labeled pairs than Clopidogrel

SPL labels Repaglinide + Clopidogrel as minor; Repaglinide 17 / Clopidogrel 10 in that band.

Mechanism on file: Clopidogrel blocks the enzyme that breaks down repaglinide. This causes repaglinide levels to rise much higher than normal in your blood.

FDA SPL severity: Minor

Repaglinide

Full Repaglinide label record

Meglitinide

Clopidogrel

Full Clopidogrel label record

Antiplatelet Agent

Repaglinide + Clopidogrel · SPL mechanism field

Clopidogrel blocks the enzyme that breaks down repaglinide. This causes repaglinide levels to rise much higher than normal in your blood.

Minor band excerpt · Repaglinide with Clopidogrel

( 7.7 ) Repaglinide (CYP2C8 substrates): Increases substrate plasma concentrations. 7.8 Repaglinide (CYP2C8 Substrates) The acyl-β-glucuronide metabolite of clopidogrel is a strong inhibitor of CYP2C8. Clopidogrel increased repaglinide exposures by 3.9-fold to 5.1-fold [see Clinical Pharmacology (12.3) ] .

Repaglinide · 2 major-labeled pairs (vs Clopidogrel's 0)

View all Repaglinide interactions →

FDA Drug Labels (SPL) via openFDA. Registry display only. Not medical advice.