Atovaquone/Proguanil and Warfarin Interaction

Drug interaction information between Atovaquone/Proguanil and Warfarin.

Atovaquone/Proguanil and Warfarin have a documented minor interaction in FDA labeling.

FDA drug labeling documents a minor-severity interaction between Atovaquone/Proguanil and Warfarin. This page displays the available source-record category and label text. The category is not an individual risk estimate or medication-combination direction.

Drug A

Atovaquone/Proguanil

Antimalarial Combination

Drug B

Warfarin

Vitamin K Antagonist (Anticoagulant)

How They Interact

Proguanil can increase the blood-thinning effects of warfarin, which may make you bleed more easily.

FDA Label Information

( 7.1 ) • Proguanil may potentiate anticoagulant effect of warfarin and other coumarin-based anticoagulants. 7.2 Anticoagulants Proguanil may potentiate the anticoagulant effect of warfarin and other coumarin-based anticoagulants.

Atovaquone/Proguanil Also Interacts With

View all Atovaquone/Proguanil interactions →

Warfarin Also Interacts With

View all Warfarin interactions →

Frequently Asked Questions

What SPL severity band is on file for Atovaquone/Proguanil + Warfarin?

Compiled FDA labeling labels this pair minor. That is a source-record field, not an individual medication-combination decision.

Which drug in this pair has the larger labeled-interaction portfolio?

Warfarin has 163 labeled pairs on file vs Atovaquone/Proguanil's 4. In the minor band specifically: Atovaquone/Proguanil has 3 (also Tetracycline, Metoclopramide); Warfarin has 133 (also Atorvastatin, Amlodipine, Omeprazole, Famotidine).

What mechanism field is on file for Atovaquone/Proguanil and Warfarin?

Proguanil can increase the blood-thinning effects of warfarin, which may make you bleed more easily.

Warfarin carries more major-labeled pairs than Atovaquone/Proguanil

SPL source-record counts only. This page's band is minor · classes on file: Atovaquone/Proguanil (Antimalarial Combination); Warfarin (Vitamin K Antagonist (Anticoagulant)).

Warfarin has 2 major-labeled pairs vs Atovaquone/Proguanil's 0. This page itself is in the minor band, not the major band.

Atovaquone/Proguanil

0 major · 1 moderate · 3 minor · 4 total

Warfarin

2 major · 28 moderate · 133 minor · 163 total

Sources: FDA Drug Labels (SPL) via openFDA (2026). This is for informational purposes only and is not medical advice. This registry does not provide individual medication-combination directions.