PlainMeds provides educational information only. This is not medical advice. Always consult your doctor or pharmacist.

Prescription medication · Muscle Relaxant

metaxalone

Also sold as Skelaxin. Metaxalone treats the pain and discomfort caused by muscle problems.

3,268
FDA reportsLightly reported
18
InteractionsSeveral interactions
$2.61
Generic price (NADAC)

What the data shows

metaxalone (Skelaxin) is a prescription Muscle Relaxant, among the least-reported drugs the FDA tracks (3,268 FDA reports), with 18 documented drug interactions.

Reporting volume reflects how widely a drug is used and studied, not how dangerous it is, a FAERS report documents a temporal association, never proof of cause.

metaxalone (Skelaxin) is a prescription Muscle Relaxant. Metaxalone treats the pain and discomfort caused by muscle problems.

Metaxalone is a muscle relaxant. It helps relieve discomfort from painful muscle and bone problems.

Drug Pricing (NADAC)

Generic Price

$2.61/unit

Generic Available

Yes (5 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

View Alternatives → Compare with Another Drug → Full Side Effects Report →

What it does

Metaxalone treats the pain and discomfort caused by muscle problems.

Common side effects

Drowsiness, Dizziness, Headache

Key warnings

Metaxalone can cause sleepiness.

The sections below are summarized in plain English from metaxalone's FDA-approved prescribing information. They describe what the official label says, and are not personal medical advice.

How It Works

The exact way metaxalone works is not fully known. It is thought to work by making you feel sleepy. This can help to relieve muscle pain.

How to Take It

Take one 800 mg tablet three to four times a day. You can take it with or without food. Follow your doctor's instructions carefully. Do not take more than prescribed.

This is a plain-language summary of metaxalone's FDA labeling, not individualized dosing advice. Ask a pharmacist or prescriber before changing how you take this medication.

Pregnancy & Breastfeeding

It is not known if metaxalone can harm an unborn baby. Talk to your doctor if you are pregnant, plan to become pregnant, or are breastfeeding.

This is a plain-language summary of metaxalone's FDA labeling, not individualized advice. Ask a pharmacist or prescriber about pregnancy or breastfeeding on this medication.

Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule.

This is a plain-language summary of metaxalone's FDA labeling, not individualized advice. Ask a pharmacist or prescriber what to do about your specific missed dose.

Storage

Store at room temperature, between 68ºF and 77ºF.

Side Effects (from patient reports)

Based on 3,268 FDA adverse event reports.

Most-reported reactions

Adverse reactions in FAERS for metaxalone, by number of reports

reports

What this shows Bars show how often each reaction was reported, not how likely it is to happen, a report records a temporal association, never proof that the drug caused it.

Source FDA Adverse Event Reporting System (FAERS) As of 2025

Reports over time

Adverse-event reports filed for metaxalone each year to the FDA Adverse Event Reporting System (FAERS).

0100200300400 20042007201020132016201920222025 130

Year-to-year volume tracks usage, prescribing, and scrutiny, not a change in per-patient risk. Source: FDA FAERS.

Where metaxalone sits

metaxalone has more FDA adverse-event reports than 19% of the drugs FAERS tracks. A high position reflects how widely a drug is used and watched, not how dangerous it is.

fewest reports most reports

Percentile across all drugs PlainMeds tracks by FAERS report volume. The dot is metaxalone; the line is the median (50th percentile).

FDA Adverse Event Report Analysis

Detailed analysis of 3,268 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2004–2025.

Total Reports

3,268

Reports Mentioning Death

599

18.3% of reports — not proof of cause

Hospitalization Reports

771

Top Indication

Product Used For Unknown Indication

Gender Distribution

Female 2,234 (73%)
Male 812 (27%)

Age Distribution

0–17 27
18–44 541
45–64 1,002
65–74 336
75+ 142

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 COMPLETED SUICIDE 261
3 FATIGUE 196
4 PAIN 195
5 NAUSEA 190
6 HEADACHE 166
7 TOXICITY TO VARIOUS AGENTS 163
8 FALL 161
9 DIARRHOEA 132
10 DIZZINESS 120
11 DEATH 114
12 DYSPNOEA 114
13 CHRONIC KIDNEY DISEASE 111
14 RENAL FAILURE 107
15 VOMITING 105
16 BACK PAIN 99

Reactions in Death Reports

COMPLETED SUICIDE 261
TOXICITY TO VARIOUS AGENTS 155
DEATH 113
DRUG ABUSE 54
CARDIO-RESPIRATORY ARREST 45
CARDIAC ARREST 37
OVERDOSE 34
RESPIRATORY ARREST 34
ACCIDENTAL DEATH 26
RENAL FAILURE 24

Reactions in Hospitalization Reports

FALL 60
PNEUMONIA 59
NAUSEA 54
RENAL FAILURE 52
SEROTONIN SYNDROME 50
PAIN 48
FATIGUE 47
DIARRHOEA 45
DYSPNOEA 45
DIZZINESS 43

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

Metaxalone can cause sleepiness. Do not drive or operate heavy machinery until you know how it affects you. Using metaxalone with alcohol, opioids, or other drugs that cause sleepiness can be dangerous. A potentially life-threatening condition called serotonin syndrome has been reported when metaxalone is used with certain other drugs.

Known Drug Interactions

moderate tapentadol

Examples: Selective serotonin reuptake inhibitors (SSRIs), serotonin and norepinephrine reuptake inhibitors (SNRIs), tricyclic antidepressants (TCAs), triptans, 5-HT3 receptor antagonists, drugs that affect the serotonin neurotransmitter system (e.g., mirtazapine, trazodone, tramadol), certain muscle relaxants (i.e., cyclobenzaprine, metaxalone), monoamine oxidase inhibitors (those intended to treat psychiatric disorders and also others, such as linezolid and intravenous methylene blue). Due to the risk of respiratory depression with concomitant use of skeletal muscle relaxants and...

Mechanism: Both of these medications can slow down your breathing and affect your brain's serotonin levels. Combining them makes these side effects more likely and more severe.

What to do: Your healthcare provider should monitor you closely for signs of respiratory distress. Avoid this combination unless specifically directed by your doctor.

Examples of serotonergic drugs include: selective serotonin reuptake inhibitors (SSRIs), serotonin and norepinephrine reuptake inhibitors (SNRIs), tricyclic antidepressants (TCAs), triptans, 5-HT3 receptor antagonists, opioids (particularly fentanyl, meperidine, and methadone), drugs that affect the serotonin neurotransmitter system (e.g., mirtazapine, trazodone, tramadol), monoamine oxidase (MAO) inhibitors (those intended to treat psychiatric disorders and also others, such as linezolid and intravenous methylene blue).

Mechanism: Taking these two drugs together can cause a build-up of serotonin in your body, which can be life-threatening if levels become too high.

What to do: Tell your doctor immediately if you experience shivering, sweating, or a very high fever while taking these medications.

Examples of serotonergic drugs include: selective serotonin reuptake inhibitors (SSRIs), serotonin and norepinephrine reuptake inhibitors (SNRIs), tricyclic antidepressants (TCAs), triptans, 5-HT3 receptor antagonists, opioids (particularly fentanyl, meperidine, and methadone), drugs that affect the serotonin neurotransmitter system (e.g., mirtazapine, trazodone, tramadol), monoamine oxidase (MAO) inhibitors (those intended to treat psychiatric disorders and also others, such as linezolid and intravenous methylene blue).

Mechanism: Both of these drugs can increase the levels of a brain chemical called serotonin. Taking them together may cause serotonin to build up to unsafe levels in your body.

What to do: Your doctor should monitor you closely for signs of serotonin syndrome, such as confusion, sweating, or muscle stiffness.

Examples of serotonergic drugs include: selective serotonin reuptake inhibitors (SSRIs), serotonin and norepinephrine reuptake inhibitors (SNRIs), tricyclic antidepressants (TCAs), triptans, 5-HT3 receptor antagonists, opioids (particularly fentanyl, meperidine, and methadone), drugs that affect the serotonin neurotransmitter system (e.g., mirtazapine, trazodone, tramadol), monoamine oxidase (MAO) inhibitors (those intended to treat psychiatric disorders and also others, such as linezolid and intravenous methylene blue).

Mechanism: Linezolid acts as a monoamine oxidase inhibitor, which can cause serotonin levels to rise when taken with metaxalone. This combination increases the risk of a serious reaction called serotonin syndrome.

What to do: Talk to your healthcare provider about the risks, as they may need to adjust your treatment or watch for side effects.

Examples of serotonergic drugs include: selective serotonin reuptake inhibitors (SSRIs), serotonin and norepinephrine reuptake inhibitors (SNRIs), tricyclic antidepressants (TCAs), triptans, 5-HT3 receptor antagonists, opioids (particularly fentanyl, meperidine, and methadone), drugs that affect the serotonin neurotransmitter system (e.g., mirtazapine, trazodone, tramadol), monoamine oxidase (MAO) inhibitors (those intended to treat psychiatric disorders and also others, such as linezolid and intravenous methylene blue).

Mechanism: These medications both affect the chemical systems in your brain and nerves. Using them at the same time can lead to an unhealthy buildup of serotonin.

What to do: Use this combination with caution and tell your doctor immediately if you feel agitated, dizzy, or have a fast heartbeat.

Check all your medications →

This is a plain-language summary of interactions documented in FDA labeling, not individualized advice. Ask a pharmacist or prescriber before combining medications.

Common Questions

Can I drive while taking metaxalone?
Metaxalone can cause drowsiness or dizziness. Do not drive or operate heavy machinery until you know how it affects you.
Can I drink alcohol while taking metaxalone?
Drinking alcohol while taking metaxalone can increase drowsiness and other side effects. It is best to avoid alcohol.
What should I do if I experience side effects?
If you experience any bothersome or severe side effects, contact your doctor.
Can I take metaxalone with other medications?
Metaxalone can interact with other medications, especially those that cause drowsiness or affect serotonin levels. Tell your doctor about all the medications you take.
Is metaxalone addictive?
Metaxalone is not known to be addictive when taken as prescribed.
How long does it take for metaxalone to work?
Metaxalone usually starts to work within one hour. It may take a few days to feel the full effect.
Can I stop taking metaxalone suddenly?
Talk to your doctor before stopping metaxalone. Stopping suddenly may cause withdrawal symptoms.
What if the medicine doesn't seem to be working?
If your pain does not improve after a few days, contact your doctor.
Can children take metaxalone?
Metaxalone is approved for children over 12 years of age. Talk to your doctor before giving it to a child.
What are the common side effects of metaxalone?
The most commonly reported side effects of metaxalone include Drowsiness, Dizziness, Headache, Nervousness or irritability, Nausea. Based on 3,268 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
Does metaxalone interact with other medications?
Yes, metaxalone has 18 known drug interactions. Notable interactions include tapentadol, trazodone, mirtazapine. Always inform your doctor about all medications you are taking.
What drug class is metaxalone?
metaxalone belongs to the Muscle Relaxant drug class. It requires a prescription (Rx). Metaxalone treats the pain and discomfort caused by muscle problems.
Is metaxalone safe during pregnancy?
It is not known if metaxalone can harm an unborn baby. Talk to your doctor if you are pregnant, plan to become pregnant, or are breastfeeding. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

Related Medications in Muscle Relaxant

Other drugs grouped near metaxalone - same-class peers and common alternatives.

Compare metaxalone vs baclofen side-by-side →

Medication Guides

Save on metaxalone

Compare prices and find discounts at pharmacies near you. Free coupons can save up to 80% on prescriptions.

Disclosure: This link may earn us a commission at no extra cost to you. See our terms.

What the FDA Data Shows for metaxalone

The FDA label for metaxalone (sold under brand names such as Skelaxin) classifies it as a prescription-only medication in the Muscle Relaxant class. Metaxalone treats the pain and discomfort caused by muscle problems. Official labeling lists 7 commonly reported side effects, including Drowsiness, Dizziness, Headache.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 3,268 voluntary reports. The database also lists 18 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated moderate severity. NADAC pricing from CMS shows a generic unit cost of $2.61.

Report counts do not establish causation, a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice, always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: July 25, 2022

Data currency: FDA FAERS adverse-event reports through 2025, CMS NADAC acquisition-cost pricing effective December 2024, compiled and last refreshed May 2026. See our methodology for per-source dates and refresh cadence. Spot a figure that looks wrong? Report a correction.

All federal data sources used on this page