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exenatide

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Brand names: Byetta, Bydureon

GLP-1 Receptor Agonist Rx

Byetta is a medicine that helps adults with type 2 diabetes control their blood sugar. It works along with diet and exercise.

Drug Pricing (NADAC)

Brand Price

$340.29/unit

Generic Available

Yes (1 manufacturer)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

Byetta helps adults with type 2 diabetes manage their blood sugar levels.

Common side effects

Nausea, Low blood sugar, Vomiting

Key warnings

Byetta may cause serious side effects, including pancreatitis.

How It Works

Byetta is a GLP-1 receptor agonist. It works by helping your body release insulin when your blood sugar is high. It also lowers the amount of sugar your liver makes.

How to Take It

Inject Byetta under your skin within 60 minutes before your morning and evening meals. These meals should be about 6 hours apart. Start with 5 mcg twice a day. After 1 month, your doctor may increase your dose to 10 mcg twice a day.

Pregnancy & Breastfeeding

Talk to your doctor if you are pregnant or plan to become pregnant. Byetta should only be used during pregnancy if the benefit outweighs the risk to the baby. It is not known if Byetta passes into breast milk.

Missed Dose

If you miss a dose, just take your next scheduled dose as usual. Do not take an extra dose to make up for the missed one.

Storage

Store Byetta in the refrigerator. After the first use, you can keep it at room temperature for up to 30 days. Throw the pen away after 30 days, even if there is medicine left.

Side Effects (from patient reports)

Based on 64,891 FDA adverse event reports.

High blood sugar
15,473
Weight loss
12,125
Feeling sick to your stomach
12,038
Reduced appetite
5,644
Low blood sugar
5,517
Throwing up
4,345
Diarrhea
2,743
Feeling dizzy
2,671
Medicine not working
2,250
Headache
2,085

FDA Adverse Event Report Analysis

Detailed analysis of 52,302 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2005–2025.

Total Reports

52,302

Death-Related Reports

1,762

Hospitalization Reports

7,532

Top Indication

Type 2 Diabetes Mellitus

Gender Distribution

Female 32,746 (64%)
Male 18,369 (36%)

Age Distribution

0–17 50
18–44 3,015
45–64 20,550
65–74 9,220
75+ 2,393

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 BLOOD GLUCOSE INCREASED 15,472
2 WEIGHT DECREASED 12,125
3 NAUSEA 12,040
4 DECREASED APPETITE 5,643
5 BLOOD GLUCOSE DECREASED 5,517
6 VOMITING 4,345
7 DIARRHOEA 2,742
8 DIZZINESS 2,673
9 DRUG INEFFECTIVE 2,250
10 HEADACHE 2,086
11 INJECTION SITE PAIN 2,023
12 PANCREATITIS 2,012
13 INJECTION SITE BRUISING 1,843
14 INJECTION SITE HAEMORRHAGE 1,809
15 FATIGUE 1,759

Reactions in Death Reports

PANCREATIC CARCINOMA 765
DEATH 346
PANCREATIC CARCINOMA METASTATIC 268
METASTASES TO LIVER 178
RENAL FAILURE 94
PANCREATITIS 91
ADENOCARCINOMA PANCREAS 90
NAUSEA 82
WEIGHT DECREASED 77
HYPERTENSION 74

Reactions in Hospitalization Reports

WEIGHT DECREASED 1,332
NAUSEA 1,199
BLOOD GLUCOSE INCREASED 1,150
PANCREATITIS 1,033
VOMITING 813
PANCREATITIS ACUTE 574
OFF LABEL USE 550
DIARRHOEA 483
DECREASED APPETITE 481
BLOOD GLUCOSE DECREASED 431

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

Byetta may cause serious side effects, including pancreatitis. If you have severe stomach pain that won't go away, stop using Byetta and call your doctor right away. Never share your Byetta pen with anyone else, even if you change the needle.

Known Drug Interactions

Orally Administered Drugs (e.g., acetaminophen) Clinical Impact Exenatide slows gastric emptying.

Mechanism: Exenatide slows down the movement of food and medicine out of your stomach, which can delay how fast acetaminophen starts working.

What to do: You may need to change when you take your pain medicine to make sure it works effectively.

( 7 ) • Warfarin: Postmarketing reports of increased INR sometimes associated with bleeding. Warfarin Clinical Impact In a drug interaction study, BYETTA did not have a significant effect on INR [see Clinical Pharmacology (12.3) ] . There have been postmarketing reports for BYETTA of increased INR with concomitant use of warfarin, sometimes associated with bleeding [see Adverse Reactions (6.2) ] .

Mechanism: Taking these drugs together may change how your blood clots, which can lead to a higher risk of bleeding.

What to do: Your doctor should check your blood clotting tests more often if you take both of these medicines.

Common Questions

Can I use Byetta with other diabetes medicines?
Yes, but talk to your doctor about the right doses, especially if you take insulin or a sulfonylurea medicine.
What should I do if I feel sick to my stomach?
Nausea is common when starting Byetta, but it usually gets better over time. Eat smaller meals and avoid greasy foods.
Can Byetta cause low blood sugar?
Yes, especially if you are also taking insulin or a sulfonylurea. Check your blood sugar often and talk to your doctor about adjusting your doses.
Where should I inject Byetta?
You can inject it into your thigh, abdomen, or upper arm. Rotate injection sites each time.
How long does Byetta take to work?
Byetta starts working right away to help control your blood sugar after meals.
What if the Byetta solution looks cloudy?
Do not use it. The solution should be clear and colorless. Contact your pharmacist for a new pen.
Can I travel with my Byetta pen?
Yes, but keep it in its original packaging and protect it from extreme temperatures. Follow TSA guidelines.
What should I do if I have an allergic reaction?
Stop using Byetta and get medical help right away if you have hives, swelling, or trouble breathing.
Does Byetta cause weight loss?
Some people may lose weight while taking Byetta, but it is not a weight loss medicine.
Can I drink alcohol while taking Byetta?
Talk to your doctor about drinking alcohol while taking Byetta, as it can affect your blood sugar.
What are the common side effects of exenatide?
The most commonly reported side effects of exenatide include Nausea, Low blood sugar, Vomiting, Diarrhea, Feeling jittery. Based on 64,891 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
Does exenatide interact with other medications?
Yes, exenatide has 2 known drug interactions. Notable interactions include acetaminophen, warfarin. Always inform your doctor about all medications you are taking.
What drug class is exenatide?
exenatide belongs to the GLP-1 Receptor Agonist drug class. It requires a prescription (Rx). Byetta helps adults with type 2 diabetes manage their blood sugar levels.
Is exenatide safe during pregnancy?
Talk to your doctor if you are pregnant or plan to become pregnant. Byetta should only be used during pregnancy if the benefit outweighs the risk to the baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

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What the FDA Data Shows for exenatide

The FDA label for exenatide (sold under brand names such as Byetta, Bydureon) classifies it as a prescription-only medication in the GLP-1 Receptor Agonist class. Byetta helps adults with type 2 diabetes manage their blood sugar levels. Official labeling lists 10 commonly reported side effects, including Nausea, Low blood sugar, Vomiting.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 64,891 voluntary reports. The database also lists 2 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated minor severity. NADAC pricing from CMS.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: September 2, 2025

All federal data sources used on this page