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acebutolol

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Brand names: Sectral

Beta-1 Selective Blocker with ISA Rx

Acebutolol is a medicine that helps lower blood pressure and control irregular heartbeats. It belongs to a class of drugs called beta-blockers.

Drug Pricing (NADAC)

Generic Price

$0.58/unit

Generic Available

Yes (2 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

Acebutolol is used to treat high blood pressure in adults.

Common side effects

No common side effects listed.

Key warnings

You should not take acebutolol if you have a very slow heart rate, second- or third-degree heart block, heart failure, or cardiogenic shock.

How It Works

Acebutolol works by blocking the effects of certain natural chemicals in your body, like adrenaline, on the heart and blood vessels. This helps to slow down the heart rate and lower blood pressure. It also helps to make the heart beat more regularly.

How to Take It

Take acebutolol as your doctor tells you. The starting dose for high blood pressure is usually 400 mg daily. This can be taken as one dose or two divided doses. Your doctor may change your dose to find what works best for you, up to a maximum of 1200 mg per day. If you stop treatment, reduce the dosage slowly over about two weeks.

Pregnancy & Breastfeeding

Tell your doctor if you are pregnant or plan to become pregnant. It is not known if acebutolol will harm an unborn baby. Talk to your doctor about the risks and benefits of taking acebutolol while breastfeeding.

Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule.

Storage

Store acebutolol at room temperature (68° to 77°F) and protect it from light. Keep the container tightly closed.

Side Effects (from patient reports)

Based on 5,543 FDA adverse event reports.

Problems with thinking or memory
620
Falling down
615
Low blood pressure when standing up
573
Problems with balance
568
Difficulty passing stools
565
Low blood pressure
564
Feeling sleepy or drowsy
538
Difficulty moving around
508
Reduced alertness
501
Aches or soreness
491

FDA Adverse Event Report Analysis

Detailed analysis of 1,220 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2004–2025.

Total Reports

1,220

Death-Related Reports

44

Hospitalization Reports

921

Top Indication

Product Used For Unknown Indication

Gender Distribution

Female 861 (81%)
Male 207 (19%)

Age Distribution

0–17 7
18–44 16
45–64 145
65–74 115
75+ 726

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 COGNITIVE DISORDER 620
2 FALL 615
3 ORTHOSTATIC HYPOTENSION 573
4 BALANCE DISORDER 568
5 CONSTIPATION 565
6 HYPOTENSION 564
7 SEDATION 538
8 MOBILITY DECREASED 508
9 DEPRESSED LEVEL OF CONSCIOUSNESS 501
10 PAIN 491
11 SEDATION COMPLICATION 490
12 BLOOD CALCIUM DECREASED 485
13 CREATININE RENAL CLEARANCE DECREASED 485
14 TOXICITY TO VARIOUS AGENTS 473
15 DRUG INEFFECTIVE 156

Reactions in Death Reports

DRUG INTERACTION 6
HAEMATEMESIS 6
AGRANULOCYTOSIS 5
CEREBRAL HAEMATOMA 5
OFF LABEL USE 5
CONDITION AGGRAVATED 4
ACUTE KIDNEY INJURY 3
FALL 3
INTENTIONAL PRODUCT USE ISSUE 3
LEUKAEMIA 3

Reactions in Hospitalization Reports

COGNITIVE DISORDER 613
FALL 601
ORTHOSTATIC HYPOTENSION 566
BALANCE DISORDER 558
CONSTIPATION 554
HYPOTENSION 550
SEDATION 531
MOBILITY DECREASED 501
DEPRESSED LEVEL OF CONSCIOUSNESS 493
SEDATION COMPLICATION 486

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

You should not take acebutolol if you have a very slow heart rate, second- or third-degree heart block, heart failure, or cardiogenic shock.

Known Drug Interactions

7.3 Beta-Adrenergic Receptor Antagonists (e.g., acebutolol, metoprolol) Beta-adrenergic receptor antagonists have been shown to reduce the production of melatonin via specific inhibition of beta-1 adrenergic receptors.

Mechanism: Acebutolol can lower the amount of natural melatonin your body makes. This may make tasimelteon less effective since it works on the same sleep system.

What to do: Your doctor may need to monitor your sleep patterns or adjust your medications if they are not working well.

Common Questions

Can I drink alcohol while taking acebutolol?
Talk to your doctor about drinking alcohol while taking acebutolol.
Will acebutolol cure my high blood pressure?
Acebutolol helps control high blood pressure, but it is not a cure. You may need to take it for the rest of your life.
Can I stop taking acebutolol if I feel better?
Do not stop taking acebutolol without talking to your doctor. Stopping suddenly can cause serious heart problems.
Does acebutolol interact with other medications?
Yes, acebutolol can interact with other medications. Tell your doctor about all the medicines you take, including prescription and over-the-counter drugs, vitamins, and herbal supplements.
Can older patients take this medication?
Older patients may need lower doses. Doses above 800 mg/day should be avoided in the elderly.
What do I do if I think I have overdosed?
Call your doctor or seek medical attention immediately.
Can acebutolol cause weight gain?
Weight changes are not commonly reported with acebutolol.
Can acebutolol cause dizziness?
Dizziness is a possible side effect of acebutolol.
How long does it take for acebutolol to start working?
It may take a few weeks for acebutolol to fully lower your blood pressure.
What are the inactive ingredients in acebutolol?
The inactive ingredients are D&C Red 28, D&C Yellow 10, FD&C Blue 1, FD&C Red 40, gelatin, maize starch, povidone, stearic acid and titanium dioxide.
Does acebutolol interact with other medications?
Yes, acebutolol has 1 known drug interactions. Notable interactions include tasimelteon. Always inform your doctor about all medications you are taking.
What drug class is acebutolol?
acebutolol belongs to the Beta-1 Selective Blocker with ISA drug class. It requires a prescription (Rx). Acebutolol is used to treat high blood pressure in adults.
Is acebutolol safe during pregnancy?
Tell your doctor if you are pregnant or plan to become pregnant. It is not known if acebutolol will harm an unborn baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

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What the FDA Data Shows for acebutolol

The FDA label for acebutolol (sold under brand names such as Sectral) classifies it as a prescription-only medication in the Beta-1 Selective Blocker with ISA class. Acebutolol is used to treat high blood pressure in adults. Labeling covers dosing, contraindications, and monitoring requirements derived from clinical trials.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 5,543 voluntary reports. The database also lists 1 documented drug interaction derived from FDA labeling, with the top-flagged interaction rated minor severity. NADAC pricing from CMS shows a generic unit cost of $0.58.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: October 23, 2024

All federal data sources used on this page