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mexiletine Side Effects

Also known as: Mexitil

Analysis of 408 adverse event reports submitted to the FDA from 2004 to 2025.

Total Reports

408

Death-Related

75

18.4% of reports

Hospitalizations

253

62.0% of reports

Top Indication

Product Used For Unknown Indication

Most Reported Adverse Reactions

DRUG INEFFECTIVE
42
FATIGUE
31
VENTRICULAR TACHYCARDIA
31
DYSPNOEA
26
NAUSEA
24
POOR QUALITY SLEEP
24
IMPAIRED WORK ABILITY
23
IMPAIRED QUALITY OF LIFE
22
PYREXIA
22
CARDIAC FAILURE
18
HYPERTENSION
18
PNEUMONIA
18
CONTUSION
15
ALANINE AMINOTRANSFERASE INCREASED
14
CARDIAC FAILURE CONGESTIVE
14
DIARRHOEA
14
DIZZINESS
14
HERPES ZOSTER
14
RESPIRATORY FAILURE
14
CATARACT
13

Who Reports Side Effects

Gender Distribution

Female 158 (41%)
Male 230 (59%)
Unknown 1

Age Distribution

0-17 15 (5%)
18-44 24 (7%)
45-64 97 (30%)
65-74 82 (25%)
75+ 107 (33%)

Reporting Trend by Year

2004 2025

Reactions in Death Reports

Top reactions reported in 75 reports where death was an outcome. These are voluntarily reported and do not establish causation.

Reaction Reports
PNEUMONIA 11
DEATH 10
CARDIAC ARREST 8
CARDIAC FAILURE 8
NAUSEA 8
CARDIAC FAILURE CONGESTIVE 7
PAIN 7
DYSPNOEA 6
RENAL FAILURE 6
THROMBOCYTOPENIA 6
VOMITING 6
ANAEMIA 5
ANXIETY 5
ECONOMIC PROBLEM 5
GENERAL PHYSICAL HEALTH DETERIORATION 5
RESPIRATORY FAILURE 5
VENTRICULAR TACHYCARDIA 5
ASTHENIA 4
HEADACHE 4
HYPERTENSION 4

Reactions in Hospitalization Reports

Top reactions in 253 reports where hospitalization was an outcome.

Reaction Reports
FATIGUE 31
DRUG INEFFECTIVE 29
POOR QUALITY SLEEP 24
IMPAIRED WORK ABILITY 23
IMPAIRED QUALITY OF LIFE 22
DYSPNOEA 20
VENTRICULAR TACHYCARDIA 20
PYREXIA 18
HYPERTENSION 17
PNEUMONIA 15
CONTUSION 13
HERPES ZOSTER 13
NAUSEA 13
CARDIAC FAILURE 12
CARDIAC FAILURE CONGESTIVE 12
CATARACT 12
INSOMNIA 12
RESPIRATORY FAILURE 12
WEIGHT INCREASED 12
ALANINE AMINOTRANSFERASE INCREASED 11

Nearby — Related Medications

Compare mexiletine vs adenosine →

What the FAERS Data Reveals About mexiletine Side Effects

The FDA Adverse Event Reporting System (FAERS) contains 408 voluntary reports linked to mexiletine and its brand equivalents (Mexitil), spanning 2004 through 2025. Of those, 75 (18.4%) listed death as an outcome and 253 (62.0%) involved hospitalization. The most common indication reported alongside adverse events was Product Used For Unknown Indication.

Demographic breakdowns help contextualize who is being exposed to the drug. Of reports with known sex, 41% were female and 59% male; age distribution skews toward 75+, with 107 reports in that bracket. The single most reported reaction is drug ineffective with 42 submissions, followed by fatigue and ventricular tachycardia.

FAERS is a signal-detection tool, not a scorecard. Reports are voluntary, and a single case may list multiple suspect drugs, so numbers above should not be read as incidence rates or per-patient risk. Widely prescribed drugs naturally accumulate more reports than niche therapies even when individual risk is low. These aggregates are useful for spotting patterns that merit further pharmacovigilance, not for choosing between medications. This page is for educational reference only and is not medical advice — speak with a licensed clinician about any side-effect concerns.