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leuprolide Side Effects

Also known as: Lupron

Analysis of 1,385 adverse event reports submitted to the FDA from 2005 to 2025.

Total Reports

1,385

Death-Related

119

8.6% of reports

Hospitalizations

457

33.0% of reports

Top Indication

Product Used For Unknown Indication

Most Reported Adverse Reactions

DRUG INEFFECTIVE
106
FATIGUE
82
OFF LABEL USE
67
NAUSEA
61
HEADACHE
58
MALIGNANT NEOPLASM PROGRESSION
53
DISEASE PROGRESSION
50
FEBRILE NEUTROPENIA
43
PRODUCT STORAGE ERROR
41
HOT FLUSH
36
PRODUCT USE IN UNAPPROVED INDICATION
36
ANAEMIA
35
VOMITING
35
TREATMENT FAILURE
34
DIARRHOEA
33
DIZZINESS
33
ASTHENIA
32
PAIN
31
ACUTE KIDNEY INJURY
30
HYPERTENSION
30

Who Reports Side Effects

Gender Distribution

Female 555 (43%)
Male 749 (57%)

Age Distribution

0-17 90 (9%)
18-44 257 (25%)
45-64 188 (18%)
65-74 268 (26%)
75+ 243 (23%)

Reporting Trend by Year

2005 2025

Reactions in Death Reports

Top reactions reported in 119 reports where death was an outcome. These are voluntarily reported and do not establish causation.

Reaction Reports
DEATH 29
DRUG INEFFECTIVE 18
MALIGNANT NEOPLASM PROGRESSION 16
ACUTE KIDNEY INJURY 10
ANAEMIA 10
METASTASES TO BONE 9
PNEUMONIA 8
PROSTATE CANCER 8
HYPOTENSION 7
DISEASE PROGRESSION 6
FATIGUE 6
FEBRILE NEUTROPENIA 6
METASTASES TO LIVER 6
PNEUMOCYSTIS JIROVECII PNEUMONIA 6
RESPIRATORY FAILURE 6
DYSPNOEA 5
FALL 5
GASTROENTERITIS NOROVIRUS 5
OPHTHALMIC HERPES ZOSTER 5
PAIN 5

Reactions in Hospitalization Reports

Top reactions in 457 reports where hospitalization was an outcome.

Reaction Reports
FEBRILE NEUTROPENIA 37
DRUG INEFFECTIVE 35
NAUSEA 27
ACUTE KIDNEY INJURY 26
FATIGUE 26
VOMITING 24
OFF LABEL USE 23
ANAEMIA 22
FALL 20
HYPOTENSION 19
THROMBOCYTOPENIA 19
MALIGNANT NEOPLASM PROGRESSION 18
ASTHENIA 17
DRUG DEPENDENCE 17
DYSPNOEA 17
HYPERTENSION 17
INTENTIONAL PRODUCT MISUSE 17
RESPIRATORY DEPRESSION 17
DIARRHOEA 16
PNEUMOCYSTIS JIROVECII PNEUMONIA 16

Nearby — Related Medications

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What the FAERS Data Reveals About leuprolide Side Effects

The FDA Adverse Event Reporting System (FAERS) contains 1,385 voluntary reports linked to leuprolide and its brand equivalents (Lupron), spanning 2005 through 2025. Of those, 119 (8.6%) listed death as an outcome and 457 (33.0%) involved hospitalization. The most common indication reported alongside adverse events was Product Used For Unknown Indication.

Demographic breakdowns help contextualize who is being exposed to the drug. Of reports with known sex, 43% were female and 57% male; age distribution skews toward 65-74, with 268 reports in that bracket. The single most reported reaction is drug ineffective with 106 submissions, followed by fatigue and off label use.

FAERS is a signal-detection tool, not a scorecard. Reports are voluntary, and a single case may list multiple suspect drugs, so numbers above should not be read as incidence rates or per-patient risk. Widely prescribed drugs naturally accumulate more reports than niche therapies even when individual risk is low. These aggregates are useful for spotting patterns that merit further pharmacovigilance, not for choosing between medications. This page is for educational reference only and is not medical advice — speak with a licensed clinician about any side-effect concerns.