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timolol

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Brand names: Timoptic

Beta-Blocker (Ophthalmic) Rx

Timolol (Timoptic) eye drops help lower pressure inside the eye. It is used for people with glaucoma or high eye pressure.

Drug Pricing (NADAC)

Brand Price

$10.21/unit

Generic Price

$23.09/unit

Generic Available

Yes (22 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

This medicine treats high pressure inside your eye.

Common side effects

Bitter, sour, or unusual taste, Eye burning or stinging, Redness of the eye

Key warnings

Timolol can cause serious breathing problems, including asthma.

How It Works

Timolol contains two medicines that lower eye pressure. One medicine lowers the amount of fluid your eye makes. The other medicine helps fluid drain better from your eye.

How to Take It

Use one drop in the affected eye(s) two times each day. Try to use the drops about 12 hours apart. If you use other eye drops, wait at least 5 minutes before using them. This helps each medicine work correctly.

Pregnancy & Breastfeeding

Tell your doctor if you are pregnant or plan to become pregnant. This medicine should only be used during pregnancy if the benefit outweighs the risk to the baby. Timolol can pass into breast milk. Talk to your doctor about whether to stop breastfeeding or stop using this medicine.

Missed Dose

If you miss a dose, use it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule.

Storage

Store Timolol at room temperature, away from light.

Side Effects (from patient reports)

Based on 6,980 FDA adverse event reports.

The medicine did not work
3,042
The medicine did not work
783
Feeling tired
470
Allergic reaction
456
Feeling lightheaded
401
Loose stools
396
Using the medicine for something not approved
395
Difficulty breathing
363
Feeling sick to your stomach
347
Eye feels sore
327

FDA Adverse Event Report Analysis

Detailed analysis of 11,690 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2003–2025.

Total Reports

11,690

Death-Related Reports

550

Hospitalization Reports

2,304

Top Indication

Product Used For Unknown Indication

Gender Distribution

Female 6,465 (59%)
Male 4,547 (41%)

Age Distribution

0–17 130
18–44 267
45–64 1,109
65–74 1,547
75+ 2,527

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 TREATMENT FAILURE 3,042
2 DRUG INEFFECTIVE 783
3 FATIGUE 470
4 HYPERSENSITIVITY 456
5 DIZZINESS 401
6 DIARRHOEA 396
7 OFF LABEL USE 395
8 DYSPNOEA 363
9 NAUSEA 347
10 EYE IRRITATION 327
11 FALL 317
12 HEADACHE 301
13 EYE PAIN 279
14 VISION BLURRED 274
15 INTRAOCULAR PRESSURE INCREASED 272

Reactions in Death Reports

DEATH 239
DIARRHOEA 35
FALL 31
PNEUMONIA 28
RENAL FAILURE 26
SEPSIS 23
RESPIRATORY FAILURE 22
ACUTE KIDNEY INJURY 21
ASTHENIA 21
OFF LABEL USE 21

Reactions in Hospitalization Reports

DYSPNOEA 178
DIARRHOEA 161
FALL 157
FATIGUE 141
PNEUMONIA 137
ACUTE KIDNEY INJURY 132
ANAEMIA 104
BRADYCARDIA 104
DIZZINESS 103
ASTHENIA 101

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

Timolol can cause serious breathing problems, including asthma. It can also cause heart failure. If you have asthma, COPD, or heart problems, talk to your doctor before using this medicine. This medicine contains a sulfonamide and can cause a severe allergic reaction. Stop using this medicine and contact your doctor immediately if you experience any signs of an allergic reaction.

Known Drug Interactions

moderate dorzolamide

7 DRUG INTERACTIONS Potential additive effect of oral carbonic anhydrase inhibitor with dorzolamide hydrochloride and timolol maleate ophthalmic solution. ( 7.7 ) 7.1 Oral Carbonic Anhydrase Inhibitors There is a potential for an additive effect on the known systemic effects of carbonic anhydrase inhibition in patients receiving an oral carbonic anhydrase inhibitor and dorzolamide hydrochloride and timolol maleate ophthalmic solution. The concomitant administration of dorzolamide hydrochloride and timolol maleate ophthalmic solution and oral carbonic anhydrase inhibitors is not recommended.

Mechanism: Using these drugs together can cause their effects to stack up, which may lead to more side effects throughout your body.

What to do: This combination is not recommended, and you should talk to your doctor about other options.

7.8 Clonidine Oral beta-adrenergic blocking agents may exacerbate the rebound hypertension which can follow the withdrawal of clonidine.

Mechanism: Timolol is a beta-blocker that can make blood pressure rise even higher if you suddenly stop taking clonidine. This happens because the two drugs affect the nervous system's control of blood pressure in opposite ways.

What to do: If you need to stop taking clonidine, your doctor should monitor your blood pressure closely and may need to adjust your timolol dose.

7.7 CYP2D6 Inhibitors Potentiated systemic beta-blockade (e.g., decreased heart rate, depression) has been reported during combined treatment with CYP2D6 inhibitors (e.g., quinidine, SSRIs) and timolol.

Mechanism: Certain medicines can block the body from breaking down timolol. This can lead to higher levels of the drug in your system, which may cause a slow heart rate or feelings of depression.

What to do: Your doctor should monitor you for a slow pulse or mood changes if you take these medications together.

carvedilol, metoprolol, timolol ↑ beta-blockers Clinical monitoring of patients is recommended.

Mechanism: Darunavir prevents the body from clearing timolol quickly, which can cause the beta-blocker to build up to higher levels.

What to do: Your healthcare provider should monitor you for signs of a slow heart rate or low blood pressure.

7.7 CYP2D6 Inhibitors Potentiated systemic beta-blockade (e.g., decreased heart rate, depression) has been reported during combined treatment with CYP2D6 inhibitors (e.g., quinidine, SSRIs) and timolol. There have been no reports of exacerbation of rebound hypertension with ophthalmic timolol maleate.

Mechanism: Using two medications that both contain timolol can lead to an overdose, which may slow your heart rate down too much or cause low blood pressure.

What to do: Tell your doctor about all the eye drops and heart medicines you use to avoid taking too much of the same active ingredient.

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Common Questions

Can I use Timolol with other eye drops?
Yes, but wait at least 5 minutes between using Timolol and any other eye drops.
What if my eye gets irritated?
Some eye irritation is common. If it gets severe or doesn't go away, contact your doctor.
Can I wear contact lenses while using Timolol?
Ask your doctor if it is okay to wear contact lenses while using this medicine.
How long does it take for Timolol to work?
It may take a few weeks to see the full effect. Keep using the drops as prescribed.
What should I do if I experience dizziness?
If you feel dizzy, sit or lie down until it passes. Avoid driving or operating machinery.
Can Timolol affect my heart?
Yes, Timolol can affect your heart. Tell your doctor if you have heart problems.
Is it okay to drive after using the drops?
Your vision may be blurred temporarily after using the drops. Wait until your vision is clear before driving.
What if I accidentally use too many drops?
Using too many drops is unlikely to cause serious problems. However, contact your doctor if you are concerned.
Can I stop using Timolol if my eye pressure is better?
Do not stop using Timolol without talking to your doctor first. Your eye pressure may increase if you stop suddenly.
Does this medicine have preservatives?
Yes, this medicine contains benzalkonium chloride as a preservative.
What are the common side effects of timolol?
The most commonly reported side effects of timolol include Bitter, sour, or unusual taste, Eye burning or stinging, Redness of the eye, Blurred vision, Eye itching. Based on 6,980 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
Does timolol interact with other medications?
Yes, timolol has 6 known drug interactions. Notable interactions include dorzolamide, clonidine, brimonidine/timolol. Always inform your doctor about all medications you are taking.
What drug class is timolol?
timolol belongs to the Beta-Blocker (Ophthalmic) drug class. It requires a prescription (Rx). This medicine treats high pressure inside your eye.
Is timolol safe during pregnancy?
Tell your doctor if you are pregnant or plan to become pregnant. This medicine should only be used during pregnancy if the benefit outweighs the risk to the baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.
Has timolol been recalled?
There are 6 recalls associated with timolol products. Lack of Assurance of Sterility; atypical weight loss due to improper bottle sealing leading to potential sterility concerns. Check the recalls section below for full details and affected products.

Active Recalls

Class II September 5, 2025

Lack of Assurance of Sterility; atypical weight loss due to improper bottle sealing leading to potential sterility concerns

Apotex Corp.

Class II July 5, 2025

Defective Container: spike of the cap becomes lodged in the nozzle of the product bottle.

FDC Limited

Class II April 18, 2025

Defective Container: Unable to get the solution out of the bottle as the spike of the cap was lodged in the nozzle of the product bottle.

FDC Limited

Class II October 29, 2024

Defective Container: Unable to get the solution out of the bottle as the spike of the cap was lodged in the nozzle of the product bottle

FDC Limited

Class II August 12, 2024

Defective Container: patients are unable to get the solution out of the bottle as the spike of the cap was lodged in the nozzle of the product bottle.

FDC Limited

Class III August 8, 2022

Identification of an unknown impurity at the 12-month stability point. Further investigation has identified the impurity as Timolol Phenol S-Oxide.

Akorn, Inc

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What the FDA Data Shows for timolol

The FDA label for timolol (sold under brand names such as Timoptic) classifies it as a prescription-only medication in the Beta-Blocker (Ophthalmic) class. This medicine treats high pressure inside your eye. Official labeling lists 5 commonly reported side effects, including Bitter, sour, or unusual taste, Eye burning or stinging, Redness of the eye.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 6,980 voluntary reports. The database also lists 6 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated moderate severity. NADAC pricing from CMS shows a generic unit cost of $23.09 versus $10.21 for the brand.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history (currently 6 recall records on file), and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: December 22, 2025

All federal data sources used on this page