PlainMeds provides educational information only. This is not medical advice. Always consult your doctor or pharmacist.

linaclotide

Verify with FDA → · CMS NADAC pricing →

Brand names: Linzess

Guanylate Cyclase-C Agonist Rx

Linzess is a medicine that helps treat certain bowel problems. It works by helping your bowels move more regularly.

Drug Pricing (NADAC)

Brand Price

$17.30/unit

Generic Available

No

ABBVIE

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

Linzess is used to treat irritable bowel syndrome with constipation (IBS-C) in adults and children ages 7 and older.

Common side effects

Diarrhea, Abdominal pain, Gas

Key warnings

Linzess can cause serious dehydration in children under 2 years old.

How It Works

Linzess is a guanylate cyclase-C agonist. It works by increasing fluid in your intestines. This helps to soften stool and make bowel movements easier.

How to Take It

Take Linzess on an empty stomach, at least 30 minutes before a meal. Try to take it around the same time each day. Swallow the capsule whole; do not crush or chew it. If you have trouble swallowing, you can open the capsule and mix the contents with applesauce or water.

Pregnancy & Breastfeeding

It is not expected that Linzess will harm your unborn baby. Linaclotide was not found in breast milk, so it is not expected to harm a breastfeeding baby.

Missed Dose

If you miss a dose, skip it and take your next dose at the regular time. Do not take two doses at the same time.

Storage

Store Linzess at room temperature (between 59°F and 86°F) in its original container, protected from moisture.

Side Effects (from patient reports)

Based on 20,416 FDA adverse event reports.

Diarrhea
4,502
The medicine is not working
4,365
Using the medicine for something it's not approved for
3,216
Constipation
1,862
Feeling sick to your stomach
1,373
Feeling tired
1,111
Bloating
1,100
Stomach pain
1,009
Headache
982
Pain
896

FDA Adverse Event Report Analysis

Detailed analysis of 24,979 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2012–2025.

Total Reports

24,979

Death-Related Reports

988

Hospitalization Reports

3,610

Top Indication

Product Used For Unknown Indication

Gender Distribution

Female 16,594 (73%)
Male 6,185 (27%)

Age Distribution

0–17 310
18–44 1,604
45–64 4,111
65–74 2,676
75+ 2,808

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 DIARRHOEA 4,502
2 DRUG INEFFECTIVE 4,365
3 OFF LABEL USE 3,216
4 CONSTIPATION 1,862
5 NAUSEA 1,373
6 FATIGUE 1,111
7 ABDOMINAL DISTENSION 1,100
8 ABDOMINAL PAIN 1,009
9 HEADACHE 982
10 PAIN 896
11 ABDOMINAL PAIN UPPER 884
12 DIZZINESS 796
13 INAPPROPRIATE SCHEDULE OF PRODUCT ADMINISTRATION 727
14 FLATULENCE 675
15 FALL 648

Reactions in Death Reports

DEATH 479
COMPLETED SUICIDE 93
CARDIAC ARREST 71
FALL 39
TOXICITY TO VARIOUS AGENTS 35
CHRONIC KIDNEY DISEASE 33
PNEUMONIA 32
ACUTE KIDNEY INJURY 31
CONSTIPATION 31
CARDIO-RESPIRATORY ARREST 30

Reactions in Hospitalization Reports

FALL 335
CONSTIPATION 330
NAUSEA 319
DIARRHOEA 310
PNEUMONIA 249
FATIGUE 233
DYSPNOEA 231
PAIN 229
VOMITING 209
OFF LABEL USE 204

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

Linzess can cause serious dehydration in children under 2 years old. Do not give Linzess to children under 2 years old. It is also not for people with a known or suspected blockage in their intestines.

Common Questions

Can I crush or chew the Linzess capsule?
No, do not crush or chew the Linzess capsule. Swallow it whole.
What should I do if I have severe diarrhea while taking Linzess?
Stop taking Linzess and drink plenty of fluids to rehydrate.
Can I take Linzess with food?
No, take Linzess on an empty stomach, at least 30 minutes before a meal.
Is Linzess safe to use during pregnancy?
It is not expected that Linzess will harm your unborn baby.
Can I give Linzess to my child?
Linzess can be given to children 6 years and older for certain conditions. Do not give to children under 2.
What if I can't swallow the capsule?
You can open the capsule and mix the contents with applesauce or water.
How long does it take for Linzess to work?
Linzess may start working within a few days, but it can take up to two weeks to see the full effect.
Can I take Linzess if I have a bowel obstruction?
No, you should not take Linzess if you have a known or suspected bowel obstruction.
What are the most common side effects of Linzess?
The most common side effects are diarrhea, abdominal pain, gas, and bloating.
How should I store Linzess?
Store Linzess at room temperature in its original container, protected from moisture.
What are the common side effects of linaclotide?
The most commonly reported side effects of linaclotide include Diarrhea, Abdominal pain, Gas, Bloating, Viral gastroenteritis. Based on 20,416 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
What drug class is linaclotide?
linaclotide belongs to the Guanylate Cyclase-C Agonist drug class. It requires a prescription (Rx). Linzess is used to treat irritable bowel syndrome with constipation (IBS-C) in adults and children ages 7 and older.
Is linaclotide safe during pregnancy?
It is not expected that Linzess will harm your unborn baby. Linaclotide was not found in breast milk, so it is not expected to harm a breastfeeding baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

Related Medications in Guanylate Cyclase-C Agonist

Other drugs grouped near linaclotide — same-class peers and common alternatives.

Compare linaclotide vs alosetron side-by-side →

Medication Guides

Related Health & Safety Data

Save on linaclotide

Compare prices and find discounts at pharmacies near you. Free coupons can save up to 80% on prescriptions.

Disclosure: This link may earn us a commission at no extra cost to you. See our terms.

What the FDA Data Shows for linaclotide

The FDA label for linaclotide (sold under brand names such as Linzess) classifies it as a prescription-only medication in the Guanylate Cyclase-C Agonist class. Linzess is used to treat irritable bowel syndrome with constipation (IBS-C) in adults and children ages 7 and older. Official labeling lists 6 commonly reported side effects, including Diarrhea, Abdominal pain, Gas.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 20,416 voluntary reports. Interaction data is drawn directly from FDA-approved prescribing information. NADAC pricing from CMS.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: November 4, 2025

All federal data sources used on this page