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insulin degludec

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Brand names: Tresiba

Ultra-Long-Acting Insulin Rx

Xultophy 100/3.6 is a combination of two medicines, insulin degludec and liraglutide. It helps control blood sugar in adults with type 2 diabetes, along with diet and exercise.

Drug Pricing (NADAC)

Brand Price

$32.52/unit

Generic Price

$11.39/unit

Generic Savings

65%

Generic Available

Yes (0 manufacturers)

Pricing data from NADAC (CMS), effective December 18, 2024. Compare all drug costs →

What it does

Xultophy 100/3.

Common side effects

Common cold, Headache, Feeling sick to your stomach

Key warnings

Xultophy 100/3.

How It Works

This medicine contains insulin degludec, which is a long-acting form of insulin that helps lower blood sugar levels. It also contains liraglutide, which is a GLP-1 receptor agonist. Liraglutide works by helping your body release insulin when your blood sugar is high and by slowing down the emptying of food from your stomach.

How to Take It

Inject Xultophy 100/3.6 once a day at the same time each day. You can take it with or without food. The pen delivers doses from 10 to 50 units per injection. The maximum daily dose is 50 units. Inject it under the skin of your thigh, upper arm, or abdomen, and rotate injection sites.

Pregnancy & Breastfeeding

Xultophy 100/3.6 should only be used during pregnancy if the benefit outweighs the risk to the baby. Animal studies with liraglutide, one of the medicines in this drug, have shown risks to the fetus. Talk to your doctor if you are pregnant or plan to become pregnant.

Missed Dose

If you miss a dose of Xultophy 100/3.6, take it as soon as you remember. However, do not take a double dose to make up for the missed dose.

Storage

Before first use, store Xultophy 100/3.6 in the refrigerator between 36°F to 46°F (2°C to 8°C). After first use, you can store the pen at room temperature (59°F to 86°F) or in the refrigerator for up to 21 days.

Side Effects (from patient reports)

Based on 12,391 FDA adverse event reports.

High blood sugar
3,617
Feeling sick to your stomach
1,381
Low blood sugar
1,252
The medicine is not working
963
Using the medicine for a purpose it's not approved for
901
Throwing up
894
Low blood sugar
886
Diarrhea
876
Tiredness
861
Difficulty breathing
760

FDA Adverse Event Report Analysis

Detailed analysis of 22,011 reports from the FDA Adverse Event Reporting System (FAERS). Reports span 2011–2025.

Total Reports

22,011

Death-Related Reports

1,194

Hospitalization Reports

6,329

Top Indication

Product Used For Unknown Indication

Gender Distribution

Female 11,845 (57%)
Male 9,022 (43%)

Age Distribution

0–17 334
18–44 1,396
45–64 4,924
65–74 4,036
75+ 3,041

Most Reported Adverse Reactions (FAERS)

# Reaction Reports
1 BLOOD GLUCOSE INCREASED 3,617
2 NAUSEA 1,381
3 BLOOD GLUCOSE DECREASED 1,252
4 DRUG INEFFECTIVE 963
5 OFF LABEL USE 901
6 VOMITING 894
7 HYPOGLYCAEMIA 886
8 DIARRHOEA 876
9 FATIGUE 861
10 DYSPNOEA 760
11 FALL 673
12 DIZZINESS 652
13 HEADACHE 634
14 CONSTIPATION 623
15 MALAISE 549

Reactions in Death Reports

DEATH 447
SEPSIS 265
MULTIPLE ORGAN DYSFUNCTION SYNDROME 253
GENERAL PHYSICAL HEALTH DETERIORATION 248
VOMITING 248
ASCITES 245
NAUSEA 243
HYPONATRAEMIA 241
CONSTIPATION 237
CARDIOGENIC SHOCK 236

Reactions in Hospitalization Reports

BLOOD GLUCOSE INCREASED 512
NAUSEA 453
VOMITING 423
HYPOGLYCAEMIA 409
OFF LABEL USE 341
FALL 336
DIABETIC KETOACIDOSIS 334
DYSPNOEA 316
PNEUMONIA 302
DIARRHOEA 286

Source: FDA FAERS (Adverse Event Reporting System) FDA FAERS (Adverse Event Reporting System) Reports are voluntary and do not establish causation

Serious Warnings

Xultophy 100/3.6 may increase your risk of thyroid C-cell tumors. Liraglutide, one of the medicines in Xultophy 100/3.6, caused these tumors in animals. It is not known if Xultophy 100/3.6 causes thyroid tumors in humans. You should not take this medicine if you have a personal or family history of medullary thyroid carcinoma (MTC) or if you have Multiple Endocrine Neoplasia syndrome type 2 (MEN 2). Tell your doctor if you notice a lump in your neck, have trouble swallowing or breathing, or if your voice becomes hoarse.

Known Drug Interactions

moderate fluoxetine

Drugs That May Increase the Risk of Hypoglycemia Drugs: Antidiabetic agents, ACE inhibitors, angiotensin II receptor blocking agents, disopyramide, fibrates, fluoxetine, monoamine oxidase inhibitors, pentoxifylline, pramlintide, salicylates, somatostatin analogs (e.g., octreotide), and sulfonamide antibiotics Intervention: Dosage reductions and increased frequency of glucose monitoring may be required when XULTOPHY 100/3.6 is coadministered with these drugs.

Mechanism: Fluoxetine can increase the effect of insulin, which makes your blood sugar more likely to drop to unsafe levels.

What to do: Check your blood sugar more often and talk to your doctor about adjusting your insulin dose.

moderate liraglutide

7.2 Effects of Delayed Gastric Emptying on Oral Medications Liraglutide-containing products, including XULTOPHY 100/3.6, cause a delay of gastric emptying, and thereby have the potential to impact the absorption of concomitantly administered oral medications. In clinical pharmacology trials, liraglutide did not affect the absorption of the tested orally administered medications to any clinically relevant degree [see Clinical Pharmacology ( 12.3 )] . Nonetheless, caution should be exercised when oral medications are concomitantly administered with liraglutide containing products.

Mechanism: Liraglutide slows down the movement of food and medicine through your stomach, which can change how your body absorbs pills.

What to do: Be careful when taking oral medicines with this drug and watch for changes in how well your other medicines work.

moderate pramlintide

Drugs That May Increase the Risk of Hypoglycemia Drugs: Antidiabetic agents, ACE inhibitors, angiotensin II receptor blocking agents, disopyramide, fibrates, fluoxetine, monoamine oxidase inhibitors, pentoxifylline, pramlintide, salicylates, somatostatin analogs (e.g., octreotide), and sulfonamide antibiotics Intervention: Dosage reductions and increased frequency of glucose monitoring may be required when XULTOPHY 100/3.6 is coadministered with these drugs.

Mechanism: Both drugs work to lower blood sugar, so taking them at the same time can cause your blood sugar to drop too low.

What to do: You should monitor your blood sugar levels closely and your doctor may need to lower your insulin dose.

moderate octreotide

Drugs That May Increase the Risk of Hypoglycemia Drugs: Antidiabetic agents, ACE inhibitors, angiotensin II receptor blocking agents, disopyramide, fibrates, fluoxetine, monoamine oxidase inhibitors, pentoxifylline, pramlintide, salicylates, somatostatin analogs (e.g., octreotide), and sulfonamide antibiotics Intervention: Dosage reductions and increased frequency of glucose monitoring may be required when XULTOPHY 100/3.6 is coadministered with these drugs.

Mechanism: This medication can make your body more sensitive to insulin, which increases the risk of having low blood sugar.

What to do: Your doctor may need to lower your insulin dose, and you should check your blood sugar more frequently.

Drugs That May Decrease the Blood Glucose Lowering Effect of XULTOPHY 100/3.6 Drugs: Atypical antipsychotics (e.g., olanzapine and clozapine), corticosteroids, danazol, diuretics, estrogens, glucagon, isoniazid, niacin, oral contraceptives, phenothiazines, progestogens (e.g., in oral contraceptives), protease inhibitors, somatropin, sympathomimetic agents (e.g., albuterol, epinephrine, terbutaline), and thyroid hormones.

Mechanism: Albuterol can decrease the blood-sugar-lowering effect of insulin. This can lead to higher blood sugar levels while you are using the medication.

What to do: Monitor your blood sugar levels closely if you are using albuterol. Your healthcare provider may need to adjust your insulin dose.

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Common Questions

What should I do if I experience symptoms of a thyroid tumor?
Contact your doctor immediately if you experience symptoms such as a lump in your neck, difficulty swallowing, trouble breathing, or a persistent hoarse voice.
Can I use Xultophy 100/3.6 if I have a history of pancreatitis?
Tell your doctor if you have a history of pancreatitis. If you develop symptoms of pancreatitis, such as severe abdominal pain, stop taking Xultophy 100/3.6 and contact your doctor immediately.
What should I do if I experience symptoms of low blood sugar?
If you experience symptoms of low blood sugar, such as sweating, shaking, dizziness, or confusion, treat it immediately by consuming a source of sugar, such as glucose tablets or juice. Contact your doctor if you have frequent episodes of low blood sugar.
Can I share my Xultophy 100/3.6 pen with others?
No, never share your Xultophy 100/3.6 pen with anyone else, even if the needle is changed. Sharing pens can spread infections.
What if I accidentally inject too much Xultophy 100/3.6?
If you inject too much Xultophy 100/3.6, you may experience low blood sugar. Treat it immediately by consuming a source of sugar. Contact your doctor or seek medical attention if your low blood sugar is severe or persistent.
Can other medications affect Xultophy 100/3.6?
Yes, many medications can affect blood sugar levels and may require a dosage adjustment of Xultophy 100/3.6. Tell your doctor about all the medications you are taking, including prescription and over-the-counter drugs, vitamins, and herbal supplements.
How do I dispose of used Xultophy 100/3.6 pens and needles?
Dispose of used Xultophy 100/3.6 pens and needles in a sharps container. Do not throw them in the regular trash. Ask your doctor or pharmacist for information on how to obtain a sharps container and how to dispose of it properly.
Can Xultophy 100/3.6 cause kidney problems?
Xultophy 100/3.6 can sometimes lead to dehydration, which can cause kidney problems. Drink plenty of fluids while taking this medication. Contact your doctor if you experience symptoms of dehydration, such as decreased urination, dizziness, or thirst.
What are the symptoms of a serious allergic reaction?
Symptoms of a serious allergic reaction may include rash, itching, swelling, trouble breathing, or dizziness. If you experience any of these symptoms, seek immediate medical attention.
Does Xultophy 100/3.6 have to be refrigerated?
Before you use a pen for the first time, keep it in the refrigerator. After you start using it, you can keep it at room temperature or in the refrigerator for up to 21 days.
What are the common side effects of insulin degludec?
The most commonly reported side effects of insulin degludec include Common cold, Headache, Feeling sick to your stomach, Diarrhea, Increased lipase (an enzyme). Based on 12,391 FDA adverse event reports. Always consult your healthcare provider about potential side effects.
Does insulin degludec interact with other medications?
Yes, insulin degludec has 12 known drug interactions. Notable interactions include fluoxetine, liraglutide, pramlintide. Always inform your doctor about all medications you are taking.
What drug class is insulin degludec?
insulin degludec belongs to the Ultra-Long-Acting Insulin drug class. It requires a prescription (Rx). Xultophy 100/3.
Is there a generic version of insulin degludec?
Yes, generic insulin degludec is available. The generic costs $11.39 per unit compared to $32.52 for the brand version, saving approximately 65%. Pricing is based on NADAC (National Average Drug Acquisition Cost) data from CMS.
Is insulin degludec safe during pregnancy?
Xultophy 100/3.6 should only be used during pregnancy if the benefit outweighs the risk to the baby. Always consult your healthcare provider before using any medication during pregnancy or breastfeeding.

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What the FDA Data Shows for insulin degludec

The FDA label for insulin degludec (sold under brand names such as Tresiba) classifies it as a prescription-only medication in the Ultra-Long-Acting Insulin class. Xultophy 100/3. Official labeling lists 6 commonly reported side effects, including Common cold, Headache, Feeling sick to your stomach.

Post-market surveillance from the FDA Adverse Event Reporting System (FAERS) captures real-world experience. For this drug, FAERS contains 12,391 voluntary reports. The database also lists 12 documented drug interactions derived from FDA labeling, with the top-flagged interaction rated moderate severity. NADAC pricing from CMS shows a generic unit cost of $11.39 versus $32.52 for the brand — a 65% generic savings.

Report counts do not establish causation — a FAERS entry documents a temporal association, not proof that the drug produced the outcome. Widely prescribed medications naturally accumulate more reports than niche therapies, so raw totals must be interpreted alongside total exposure. Shortage status, recall history, and patent information further shape supply and switching decisions. This page summarizes public FDA data for educational purposes only and is not a substitute for professional medical advice — always consult a licensed healthcare provider before starting, stopping, or changing any medication.

Data Sources

Drug labeling: FDA Drug Labels (SPL/DailyMed). Adverse events: FDA Adverse Event Reporting System (FAERS). Pricing: CMS National Average Drug Acquisition Cost (NADAC).

FAERS reports are voluntary and do not establish causation. Drug interactions are derived from FDA labeling and clinical references. Always consult a healthcare professional before making medication decisions.

Last updated: October 14, 2025

All federal data sources used on this page