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Drug side effects

lubiprostone Side Effects

The reactions most often reported to the FDA for lubiprostone (also sold as Amitiza), with demographics, serious outcomes, and reporting trends.

Data updated 2026-05-15

9,102
FAERS reports

Data from the FDA Adverse Event Reporting System (FAERS), 2006 to 2025. A FAERS report records a temporal association, not proof of cause. See our methodology for how figures are compiled and de-duplicated.

The most commonly reported side effects of lubiprostone come from 9,102 reports to the FDA, broken down here by frequency, patient demographics, and serious outcomes.

This page analyzes 9,102 reports to the FDA Adverse Event Reporting System (FAERS) for lubiprostone (Amitiza): the reactions reported most often, who reported them, serious outcomes such as hospitalization, and year-over-year trends. A FAERS report does not prove the drug caused the effect, and report volume tracks how widely a drug is used, not how likely an effect is for any one person. Educational information, not medical advice.

Total Reports

9,102

Reports Mentioning Death

927

10.2% of reports — not proof the medicine caused the death

Hospitalizations

3,000

33.0% of reports

Top Indication

Product Used For Unknown Indication

Most Reported Adverse Reactions

NAUSEA
765
DYSPNOEA
621
DIARRHOEA
581
CONSTIPATION
558
FATIGUE
519
HEADACHE
483
PAIN
483
DIZZINESS
440
FALL
398
VOMITING
381
CHRONIC KIDNEY DISEASE
334
MALAISE
312
PYREXIA
294
ASTHENIA
284
PNEUMONIA
277
ANXIETY
273
DECREASED APPETITE
261
RENAL FAILURE
259

Who Reports Side Effects

Gender Distribution

Female 5,912 (70%)
Male 2,538 (30%)
Unknown 35

Age Distribution

0-17 171 (3%)
18-44 891 (15%)
45-64 2,066 (35%)
65-74 1,340 (23%)
75+ 1,416 (24%)

Reporting Trend by Year

2006 2025

Reactions in Death Reports

Top reactions reported in 927 reports where death was an outcome. These are voluntarily reported and do not establish causation.

Reaction Reports
DEATH 237
PNEUMONIA 70
SEPSIS 55
MALIGNANT NEOPLASM PROGRESSION 54
CONSTIPATION 51
PYREXIA 49
DECREASED APPETITE 47
DIARRHOEA 46
RENAL FAILURE 45
INTERSTITIAL LUNG DISEASE 42
CHRONIC KIDNEY DISEASE 40
NAUSEA 36
ANAEMIA 35
ACUTE KIDNEY INJURY 34
COMPLETED SUICIDE 34
RESPIRATORY FAILURE 32
VOMITING 31
PLATELET COUNT DECREASED 30
CARDIAC FAILURE 29

Reactions in Hospitalization Reports

Top reactions in 3,000 reports where hospitalization was an outcome.

Reaction Reports
NAUSEA 246
FALL 221
DIARRHOEA 218
CONSTIPATION 217
PNEUMONIA 209
PYREXIA 182
PAIN 174
VOMITING 161
DYSPNOEA 159
FATIGUE 156
DECREASED APPETITE 142
ASTHENIA 134
DEHYDRATION 132
DIZZINESS 132
HEADACHE 128
URINARY TRACT INFECTION 128
MALAISE 126
ANXIETY 114
WEIGHT DECREASED 111

Compare lubiprostone vs alosetron →

What the FAERS Data Reveals About lubiprostone Side Effects

The FDA Adverse Event Reporting System (FAERS) contains 9,102 voluntary reports linked to lubiprostone and its brand equivalents (Amitiza), spanning 2006 through 2025. Of those, 927 (10.2%) listed death as an outcome and 3,000 (33.0%) involved hospitalization. The most common indication reported alongside adverse events was Product Used For Unknown Indication.

Demographic breakdowns help contextualize who is being exposed to the drug. Of reports with known sex, 70% were female and 30% male; age distribution skews toward 45-64, with 2,066 reports in that bracket. The single most reported reaction is nausea with 765 submissions, followed by dyspnoea and diarrhoea.

How to read these numbers

FAERS is a signal-detection tool, not a scorecard. Reports are voluntary, and a single case may list multiple suspect drugs, so numbers above should not be read as incidence rates or per-patient risk. Widely prescribed drugs naturally accumulate more reports than niche therapies even when individual risk is low. These aggregates are useful for spotting patterns that merit further pharmacovigilance, not for choosing between medications. This page is for educational reference only and is not medical advice, speak with a licensed clinician about any side-effect concerns.

Drugs With a Similar FAERS Report Volume

Other medications with a total FDA adverse-event report count closest to lubiprostone's 9,102.